PDB entry 5bx0
View 5bx0 on RCSB PDB site
Description: An Automated Microscale Thermophoresis Screening Approach for Fragment-Based Lead Discovery
Class: transferase
Keywords: fragment screening, microscale thermophoresis, transferase
Deposited on
2015-06-08, released
2015-12-23
The last revision prior to the SCOPe 2.08 freeze date was dated
2016-03-30, with a file datestamp of
2016-03-25.
Experiment type: XRAY
Resolution: 2.93 Å
R-factor: N/A
AEROSPACI score: 0.14
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dual specificity mitogen-activated protein kinase kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: MAP2K1, MEK1, PRKMK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5bx0a_ - Heterogens: 4W5
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5bx0A (A:)
gleeleldeqqrkrleafltqkqkvgelkdddfekiselgagnggvvfkvshkpsglvma
rklihleikpairnqiirelqvlhecnspyivgfygafysdgeisicmehmdggsldqvl
kkagripeqilgkvsiavikgltylrekhkimhrdvkpsnilvnsrgeiklcdfgvsgql
idsmansfvgtrsymsperlqgthysvqsdiwsmglslvemavgrypipppdakelelmf
gcqvegdaaetpprprtpgrplnkkgmdsrppmaifelldyivnepppklpsgvfslefq
dfvnkcliknpaeradlkqlmvhafikrsdaeevdfagwlcstiglnq
Sequence, based on observed residues (ATOM records): (download)
>5bx0A (A:)
eleldeqqrkrleafltqkqkvgelkdddfekiselgagnggvvfkvshkpsglvmarkl
ihleikpairnqiirelqvlhecnspyivgfygafysdgeisicmehmdggsldqvlkka
gripeqilgkvsiavikgltylrekhkimhrdvkpsnilvnsrgeiklcdfgvsgqlids
mansfvgtrsymsperlqgthysvqsdiwsmglslvemavgrypipppdakelelmfgcp
maifelldyivnepppklpsgvfslefqdfvnkcliknpaeradlkqlmvhafikrsdae
evdfagwlcstigln