PDB entry 4gpt
View 4gpt on RCSB PDB site
Description: Crystal structure of KPT251 in complex with CRM1-Ran-RanBP1
Class: protein transport/inhibitor
Keywords: HEAT repeat, protein nuclear export, KPT251, nuclear, PROTEIN TRANSPORT-INHIBITOR complex
Deposited on
2012-08-21, released
2012-09-05
The last revision prior to the SCOPe 2.02 freeze date was dated
2013-01-23, with a file datestamp of
2013-01-18.
Experiment type: XRAY
Resolution: 2.22 Å
R-factor: 0.167
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: GTP-binding nuclear protein ran
Species: Homo sapiens [TaxId:9606]
Gene: RAN, ARA24, OK/SW-cl.81
Database cross-references and differences (RAF-indexed):
- Chain 'B':
Compound: Ran-specific GTPase-activating protein 1
Species: Saccharomyces cerevisiae [TaxId:4932]
Gene: YRB1, CST20, HTN1, SFO1, YDR002W, YD8119.08
Database cross-references and differences (RAF-indexed):
- Uniprot P41920
- conflict (17)
- conflict (36)
Domains in SCOPe 2.02: d4gptb_ - Chain 'C':
Compound: Exportin-1
Species: Saccharomyces cerevisiae [TaxId:4932]
Gene: CRM1, KAP124, XPO1, YGR218W, G8514
Database cross-references and differences (RAF-indexed):
- Uniprot P30822 (2-End)
- expression tag (0-1)
- engineered mutation (540)
- engineered mutation (1023)
- Heterogens: GNP, MG, EDO, CL, 51K, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
No sequence available.
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4gptB (B:)
dihfepvvhlekvdvktaeedeevlykvraklfrfdkdakewkergtgdckflknkktnk
vrilmrrdktlkicanhiiapeytlkpnvgsdrswvyactadiaegeaeaftfairfgsk
enadkfkeefekaqeinkka
Sequence, based on observed residues (ATOM records): (download)
>4gptB (B:)
taeedeevlykvraklfrfdkdakewkergtgdckflknkktnkvrilmrrdktlkican
hiiapeytlkpnvgsdrswvyactadiaegeaeaftfairfgskenadkfkeefekaqei
nkk
- Chain 'C':
No sequence available.