PDB entry 6fa2
View 6fa2 on RCSB PDB site
Description: Antibody derived (Abd-5) small molecule binding to KRAS.
Class: oncoprotein
Keywords: Abd-5, inhibitor, KRAS, ONCOPROTEIN
Deposited on
2017-12-15, released
2018-09-05
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-09-05, with a file datestamp of
2018-08-31.
Experiment type: XRAY
Resolution: 2.6 Å
R-factor: N/A
AEROSPACI score: 0.2
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: GTPase KRas
Species: Homo sapiens [TaxId:9606]
Gene: KRAS, KRAS2, RASK2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6fa2a_ - Chain 'B':
Compound: GTPase KRas
Species: Homo sapiens [TaxId:9606]
Gene: KRAS, KRAS2, RASK2
Database cross-references and differences (RAF-indexed):
- Uniprot P01116 (3-169)
- expression tag (0-2)
- engineered mutation (63)
Domains in SCOPe 2.08: d6fa2b1, d6fa2b2 - Chain 'C':
Compound: GTPase KRas
Species: Homo sapiens [TaxId:9606]
Gene: KRAS, KRAS2, RASK2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6fa2c1, d6fa2c2 - Chain 'D':
Compound: GTPase KRas
Species: Homo sapiens [TaxId:9606]
Gene: KRAS, KRAS2, RASK2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6fa2d1, d6fa2d2 - Chain 'E':
Compound: GTPase KRas
Species: Homo sapiens [TaxId:9606]
Gene: KRAS, KRAS2, RASK2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6fa2e1, d6fa2e2 - Chain 'F':
Compound: GTPase KRas
Species: Homo sapiens [TaxId:9606]
Gene: KRAS, KRAS2, RASK2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6fa2f1, d6fa2f2 - Heterogens: MG, GNP, D2W, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>6fa2A (A:)
mteyklvvvgaggvgksaltiqliqnhfvdeydptiedsyrkqvvidgetclldildtag
heeysamrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnkcdl
psrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
- Chain 'B':
Sequence, based on SEQRES records: (download)
>6fa2B (B:)
fqgmteyklvvvgaggvgksaltiqliqnhfvdeydptiedsyrkqvvidgetclldild
tagheeysamrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnk
cdlpsrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
Sequence, based on observed residues (ATOM records): (download)
>6fa2B (B:)
fqgmteyklvvvgaggvgksaltiqliqnhfvdeydptiedsyrkqvvidgetclldild
taghesamrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnkcd
lpsrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
- Chain 'C':
Sequence, based on SEQRES records: (download)
>6fa2C (C:)
yfqgmteyklvvvgaggvgksaltiqliqnhfvdeydptiedsyrkqvvidgetclldil
dtagheeysamrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgn
kcdlpsrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
Sequence, based on observed residues (ATOM records): (download)
>6fa2C (C:)
yfqgmteyklvvvgaggvgksaltiqliqnhfvdeydptdsyrkqvvidgetclldildt
agsamrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnkcdlps
rtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
- Chain 'D':
Sequence, based on SEQRES records: (download)
>6fa2D (D:)
fqgmteyklvvvgaggvgksaltiqliqnhfvdeydptiedsyrkqvvidgetclldild
tagheeysamrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnk
cdlpsrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
Sequence, based on observed residues (ATOM records): (download)
>6fa2D (D:)
fqgmteyklvvvgaggvgksaltiqliqnhfvdeydsyrkqvvidgetclldildtagrd
qymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnkcdlpsrtvdtkq
aqdlarsygipfietsaktrqgvddafytlvreirkhk
- Chain 'E':
Sequence, based on SEQRES records: (download)
>6fa2E (E:)
fqgmteyklvvvgaggvgksaltiqliqnhfvdeydptiedsyrkqvvidgetclldild
tagheeysamrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnk
cdlpsrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
Sequence, based on observed residues (ATOM records): (download)
>6fa2E (E:)
fqgmteyklvvvgaggvgksaltiqliqnhfvdeydptiedsyrkqvvidgetclldild
tagmrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnkcdlpsr
tvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
- Chain 'F':
Sequence, based on SEQRES records: (download)
>6fa2F (F:)
fqgmteyklvvvgaggvgksaltiqliqnhfvdeydptiedsyrkqvvidgetclldild
tagheeysamrdqymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnk
cdlpsrtvdtkqaqdlarsygipfietsaktrqgvddafytlvreirkhk
Sequence, based on observed residues (ATOM records): (download)
>6fa2F (F:)
fqgmteyklvvvgaggvgksaltiqliqnhfvdedsyrkqvvidgetclldildtagmrd
qymrtgegflcvfainntksfedihhyreqikrvkdsedvpmvlvgnkcdlpsrtvdtkq
aqdlarsygipfietsaktrqgvddafytlvreirkhk