PDB entry 4xp3
View 4xp3 on RCSB PDB site
Description: Crystal structure of ERK2 in complex with an inhibitor
Class: transferase
Keywords: SERINE/THREONINE-PROTEIN KINASE, transferase
Deposited on
2015-01-16, released
2015-08-12
The last revision prior to the SCOPe 2.06 freeze date was dated
2015-08-19, with a file datestamp of
2015-08-14.
Experiment type: XRAY
Resolution: 1.78 Å
R-factor: N/A
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Mapk1, Erk2, Mapk, Prkm1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4xp3a_ - Heterogens: DX4, SO4, DMS, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4xp3A (A:)
gpemvrgqvfdvgprytnlsyigegaygmvcsaydnlnkvrvaikkispfehqtycqrtl
reikillrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyf
lyqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadpdhdhtgflteyva
trwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsq
edlnciinlkarnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqala
hpyleqyydpsdepiaeapfkfdmelddlpkeklkelifeetarfqpgyrs
Sequence, based on observed residues (ATOM records): (download)
>4xp3A (A:)
gpemvrgqvfdvgprytnlsyigegaygmvcsaydnlnkvrvaikkispfehqtycqrtl
reikillrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyf
lyqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadpdhdhtgflteyva
trwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsq
edlnciinlkarnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqala
hpyleqyydpsdepiaeapfkflpkeklkelifeetarfqp