PDB entry 4ft9
View 4ft9 on RCSB PDB site
Description: Crystal Structure of the CHK1
Class: TRANSFERASE/TRANSFERASE inhibitor
Keywords: TRANSFERASE, TRANSFERASE-TRANSFERASE inhibitor complex
Deposited on
2012-06-27, released
2012-08-22
The last revision prior to the SCOPe 2.06 freeze date was dated
2013-05-29, with a file datestamp of
2013-05-24.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: 0.163
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4ft9a_ - Heterogens: H4K, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4ft9A (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkm
lnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvyl
hgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkr
refhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplal
lhkilvenpsaritipdikkdrwynkplkkgakrprvts
Sequence, based on observed residues (ATOM records): (download)
>4ft9A (A:)
avpfvedwdlvqtlgeggevqlavnrvteeavavkivdmenikkeicinkmlnhenvvkf
yghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithrd
ikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepvd
vwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilvenp
saritipdikkdrwynkplkkgakrprvts