PDB entry 2geb
View 2geb on RCSB PDB site
Description: Crystal structure of the Thermoanaerobacter tengcongensis hypoxanthine-guanine phosphoribosyltransferase L160I mutant: insights into the inhibitor design
Class: transferase
Keywords: HGPRT, mutant, inhibitor design, selectivity, TRANSFERASE
Deposited on
2006-03-19, released
2007-04-03
The last revision prior to the SCOPe 2.07 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 1.7 Å
R-factor: 0.204
AEROSPACI score: 0.53
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: hypoxanthine-guanine phosphoribosyltransferase
Species: Thermoanaerobacter tengcongensis [TaxId:119072]
Gene: HGPRT, Hpt
Database cross-references and differences (RAF-indexed):
- GB AAM25533 (4-End)
- expression tag (0-3)
- engineered (56)
- engineered (70)
- engineered (163)
Domains in SCOPe 2.07: d2geba1, d2geba2 - Heterogens: CA, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2gebA (A:)
rgshmpspmedieeiliteeqlkakvkelgemitrdyegkdlvligvlkgaimfmsglsr
aidlplsidflavssygsstkssgivkiikdhdidiegkdvlivediidsgltlaylret
llgrkprslkictildkperreadvkvdycgfkipdkfvvgygidyaekyrnlpfigvlk
pelyk
Sequence, based on observed residues (ATOM records): (download)
>2gebA (A:)
rgshmpspmedieeiliteeqlkakvkelgemitrdyegkdlvligvlkgaimfmsglsr
aidlplsidflavssygsstkssgivkiikdhdidiegkdvlivediidsgltlaylret
llgrkprslkictildkperreadvkvdycgfkipdkfvvgygidyaekyrnlpfigvlk
pely