PDB entry 2noa
View 2noa on RCSB PDB site
Description: The structure of deoxycytidine kinase complexed with lamivudine and ADP.
Class: transferase
Keywords: dCK, 3TC, human deoxycytidine kinase, L-dC, enantiomer, antiviral, Lamivudine, Epivir, TRANSFERASE
Deposited on
2006-10-25, released
2007-02-13
The last revision prior to the SCOPe 2.06 freeze date was dated
2009-02-24, with a file datestamp of
2009-03-01.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.197
AEROSPACI score: 0.5
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Deoxycytidine kinase
Species: Homo sapiens [TaxId:9606]
Gene: DCK
Database cross-references and differences (RAF-indexed):
- Uniprot P27707 (Start-279)
- engineered (64)
- engineered (78)
- engineered (165)
Domains in SCOPe 2.06: d2noaa_ - Chain 'B':
Compound: Deoxycytidine kinase
Species: Homo sapiens [TaxId:9606]
Gene: DCK
Database cross-references and differences (RAF-indexed):
- Uniprot P27707 (Start-279)
- engineered (64)
- engineered (78)
- engineered (165)
Domains in SCOPe 2.06: d2noab_ - Heterogens: ADP, 3TC, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2noaA (A:)
mgsshhhhhhssglvprgshmatppkrsspsfsassegtrikkisiegniaagkstfvni
lkqlsedwevvpepvarwsnvqstqdefeeltmsqknggnvlqmmyekperwsftfqtya
clsriraqlaslngklkdaekpvlffersvysdryifasnlyesesmnetewtiyqdwhd
wmnnqfgqsleldgiiylqatpetclhriylrgrneeqgipleyleklhykheswllhrt
lktnfdylqevpiltldvnedfkdkyeslvekvkeflstl
Sequence, based on observed residues (ATOM records): (download)
>2noaA (A:)
trikkisiegniaagkstfvnilkqlsedwevvpepvarwsnvqstqdefeeltmsqkng
gnvlqmmyekperwsftfqtyaclsriraqlaslngklkdaekpvlffersvysdryifa
snlyesesmnetewtiyqdwhdwmnnqfgqsleldgiiylqatpetclhriylrgrneeq
gipleyleklhykheswllhrtlktnfdylqevpiltldvnedfkdkyeslvekvkefls
tl
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2noaB (B:)
mgsshhhhhhssglvprgshmatppkrsspsfsassegtrikkisiegniaagkstfvni
lkqlsedwevvpepvarwsnvqstqdefeeltmsqknggnvlqmmyekperwsftfqtya
clsriraqlaslngklkdaekpvlffersvysdryifasnlyesesmnetewtiyqdwhd
wmnnqfgqsleldgiiylqatpetclhriylrgrneeqgipleyleklhykheswllhrt
lktnfdylqevpiltldvnedfkdkyeslvekvkeflstl
Sequence, based on observed residues (ATOM records): (download)
>2noaB (B:)
rikkisiegniaagkstfvnilkqlsedwevvpepvarwsnvqggnvlqmmyekperwsf
tfqtyaclsriraqlaslngdaekpvlffersvysdryifasnlyesesmnetewtiyqd
whdwmnnqgqsleldgiiylqatpetclhriylrgrneeqgipleyleklhykheswllh
rtlktnfdylqevpiltldvnedfkdkyeslvekvkeflstl