PDB entry 6b1h
View 6b1h on RCSB PDB site
Description: Crystal structure KPC-2 beta-lactamase complexed with WCK 4234 by co-crystallization
Class: HYDROLASE/HYDROLASE Inhibitor
Keywords: Inhibitor, complex, HYDROLASE, HYDROLASE-HYDROLASE Inhibitor complex
Deposited on
2017-09-18, released
2018-08-01
The last revision prior to the SCOPe 2.07 freeze date was dated
2018-08-01, with a file datestamp of
2018-07-27.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: N/A
AEROSPACI score: 0.37
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Carbapenem-hydrolyzing beta-lactamase KPC
Species: Klebsiella pneumoniae [TaxId:573]
Gene: bla, kpc, kpc1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d6b1ha_ - Chain 'B':
Compound: Carbapenem-hydrolyzing beta-lactamase KPC
Species: Klebsiella pneumoniae [TaxId:573]
Gene: bla, kpc, kpc1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d6b1hb_ - Heterogens: C8Y, SO4, CL, ACT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>6b1hA (A:)
ataltnlvaepfakleqdfggsigvyamdtgsgatvsyraeerfplcssfkgflaaavla
rsqqqaglldtpirygknalvpwspisekylttgmtvaelsaaavqysdnaaanlllkel
ggpagltafmrsigdttfrldrwelelnsaipgdardtsspravteslqkltlgsalaap
qrqqfvdwlkgnttgnhriraavpadwavgdktgtcgvygtandyavvwptgrapivlav
ytrapnkddkhseaviaaaarlaleglg
- Chain 'B':
Sequence, based on SEQRES records: (download)
>6b1hB (B:)
ataltnlvaepfakleqdfggsigvyamdtgsgatvsyraeerfplcssfkgflaaavla
rsqqqaglldtpirygknalvpwspisekylttgmtvaelsaaavqysdnaaanlllkel
ggpagltafmrsigdttfrldrwelelnsaipgdardtsspravteslqkltlgsalaap
qrqqfvdwlkgnttgnhriraavpadwavgdktgtcgvygtandyavvwptgrapivlav
ytrapnkddkhseaviaaaarlaleglg
Sequence, based on observed residues (ATOM records): (download)
>6b1hB (B:)
ltnlvaepfakleqdfggsigvyamdtgsgatvsyraeerfplcssfkgflaaavlarsq
qqaglldtpirygknalvpwspisekylttgmtvaelsaaavqysdnaaanlllkelggp
agltafmrsigdttfrldrwelelnsaipgdardtsspravteslqkltlgsalaapqrq
qfvdwlkgnttgnhriraavpadwavgdktgtcgvygtandyavvwptgrapivlavytr
apnkddkhseaviaaaarlaleglg