PDB entry 5p9k

View 5p9k on RCSB PDB site
Description: CRYSTAL STRUCTURE OF BTK with CNX 774
Class: transferase
Keywords: lead optimization, transferase
Deposited on 2016-09-20, released 2017-05-24
The last revision prior to the SCOPe 2.07 freeze date was dated 2017-05-24, with a file datestamp of 2017-05-19.
Experiment type: XRAY
Resolution: 1.28 Å
R-factor: N/A
AEROSPACI score: 0.61 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Tyrosine-protein kinase BTK
    Species: Homo sapiens [TaxId:9606]
    Gene: BTK, AGMX1, ATK, BPK
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d5p9ka_
  • Heterogens: 7G8, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5p9kA (A:)
    gknapstaglgygsweidpkdltflkelgtgqfgvvkygkwrgqydvaikmikegsmsed
    efieeakvmmnlsheklvqlygvctkqrpifiiteymangcllnylremrhrfqtqqlle
    mckdvceameyleskqflhrdlaarnclvndqgvvkvsdfglsryvlddeytssvgskfp
    vrwsppevlmyskfssksdiwafgvlmweiyslgkmpyerftnsetaehiaqglrlyrph
    lasekvytimyscwhekaderptfkillsnildvmdees
    

    Sequence, based on observed residues (ATOM records): (download)
    >5p9kA (A:)
    glgygsweidpkdltflkelgtgqfgvvkygkwrgqydvaikmikegsmsedefieeakv
    mmnlsheklvqlygvctkqrpifiiteymangcllnylremrhrfqtqqllemckdvcea
    meyleskqflhrdlaarnclvndqgvvkvsdfglsryvlddeytssvgskfpvrwsppev
    lmyskfssksdiwafgvlmweiyslgkmpyerftnsetaehiaqglrlyrphlasekvyt
    imyscwhekaderptfkillsnildvmdees