PDB entry 5ak2
View 5ak2 on RCSB PDB site
Description: Oxyphenylpropenoic acids as Oral Selective Estrogen Receptor Down- Regulators.
Class: signaling protein
Keywords: signaling protein
Deposited on
2015-02-27, released
2015-04-22
The last revision prior to the SCOPe 2.07 freeze date was dated
2015-05-13, with a file datestamp of
2015-05-08.
Experiment type: XRAY
Resolution: 2.19 Å
R-factor: N/A
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot P03372 (20-End)
- expression tag (16-19)
- engineered mutation (94)
- engineered mutation (130)
- engineered mutation (249)
Domains in SCOPe 2.07: d5ak2a1, d5ak2a2 - Chain 'B':
Compound: Estrogen receptor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot P03372
- engineered mutation (94)
- engineered mutation (130)
Domains in SCOPe 2.07: d5ak2b_ - Heterogens: 85Z, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5ak2A (A:)
mhhhhhhgggenlyfqgshmalsltadqmvsalldaeppilyseydptrpfseasmmgll
tnladrelvhminwakrvpgfvdltlhdqvhllesawleilmiglvwrsmehpgkllfap
nllldrnqgksvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstl
ksleekdhihrvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehly
smksknvvpsydlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>5ak2A (A:)
gshmalsltadqmvsalldaeppilysesmmglltnladrelvhminwakrvpgfvdltl
hdqvhllesawleilmiglvwrsmehpgkllfapnllldrnqgksvegmveifdmllats
srfrmmnlqgeefvclksiillnsgvytsleekdhihrvldkitdtlihlmakagltlqq
qhqrlaqlllilshirhmsnkgmehlysmvpsydlllemldahrlhap
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5ak2B (B:)
mhhhhhhgggenlyfqgshmalsltadqmvsalldaeppilyseydptrpfseasmmgll
tnladrelvhminwakrvpgfvdltlhdqvhllesawleilmiglvwrsmehpgkllfap
nllldrnqgksvegmveifdmllatssrfrmmnlqgeefvclksiillnsgvytflsstl
ksleekdhihrvldkitdtlihlmakagltlqqqhqrlaqlllilshirhmsnkgmehly
smksknvvpsydlllemldahrlhapts
Sequence, based on observed residues (ATOM records): (download)
>5ak2B (B:)
lsltadqmvsalldaeppilysepfseasmmglltnladrelvhminwakrvpgfvdltl
hdqvhllesawleilmiglvwrsmehpgkllfapnllldrnqgksvegmveifdmllats
srfrmmnlqgeefvclksiillnsgvykdhihrvldkitdtlihlmakagltlqqqhqrl
aqlllilshirhmsnkgmehlysmllemld