PDB entry 6yzm
View 6yzm on RCSB PDB site
Description: Carborane nido-pentyl-sulfonamide in complex with CA IX mimic
Class: lyase
Keywords: carbonic anhydrase, ca inhibitor, lyase
Deposited on
2020-05-07, released
2020-10-28
The last revision prior to the SCOPe 2.07 freeze date was dated
2020-10-28, with a file datestamp of
2020-10-23.
Experiment type: XRAY
Resolution: 1.5 Å
R-factor: N/A
AEROSPACI score: 0.57
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Carbonic anhydrase 2
Species: Homo sapiens [TaxId:9606]
Gene: CA2
Database cross-references and differences (RAF-indexed):
- Uniprot P00918 (Start-259)
- engineered mutation (64)
- engineered mutation (66)
- engineered mutation (68)
- engineered mutation (90)
- engineered mutation (129)
- engineered mutation (168)
- engineered mutation (202)
Domains in SCOPe 2.07: d6yzma_ - Heterogens: Q4B, ZN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6yzmA (A:)
mshhwgygkhngpehwhkdfpiakgerqspvdidthtakydpslkplsvsydqatslril
nnghsfqvtfddsqdkavlkggpldgtyrllqfhfhwgsldgqgsehtvdkkkyaaelhl
vhwntkygdvgkavqqpdglavlgiflkvgsakpglqkvvdvldsiktegksadftnfdp
rgllpesldywtypgslttpplaecvtwivlkepisvsseqvlkfrklnfngegepeelm
vdnwrpaqplknrqikasfk
Sequence, based on observed residues (ATOM records): (download)
>6yzmA (A:)
hwgygkhngpehwhkdfpiakgerqspvdidthtakydpslkplsvsydqatslrilnng
hsfqvtfddsqdkavlkggpldgtyrllqfhfhwgsldgqgsehtvdkkkyaaelhlvhw
ntkygdvgkavqqpdglavlgiflkvgsakpglqkvvdvldsiktegksadftnfdprgl
lpesldywtypgslttpplaecvtwivlkepisvsseqvlkfrklnfngegepeelmvdn
wrpaqplknrqikasfk