PDB entry 5g22

View 5g22 on RCSB PDB site
Description: Plasmodium vivax N-myristoyltransferase in complex with a quinoline inhibitor (compound 26)
Class: transferase
Keywords: transferase, myristoylation, malaria, inhibitor, quinoline, drug design
Deposited on 2016-04-06, released 2017-02-15
The last revision prior to the SCOPe 2.07 freeze date was dated 2017-06-28, with a file datestamp of 2017-06-23.
Experiment type: XRAY
Resolution: 2.32 Å
R-factor: N/A
AEROSPACI score: 0.23 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Glycylpeptide N-tetradecanoyltransferase
    Species: Plasmodium vivax [TaxId:5855]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d5g22a1, d5g22a2
  • Chain 'B':
    Compound: Glycylpeptide N-tetradecanoyltransferase
    Species: Plasmodium vivax [TaxId:5855]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d5g22b1, d5g22b2
  • Chain 'C':
    Compound: Glycylpeptide N-tetradecanoyltransferase
    Species: Plasmodium vivax [TaxId:5855]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d5g22c1, d5g22c2
  • Heterogens: NHW, YN4, SO4, MG, CL, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence; same for both SEQRES and ATOM records: (download)
    >5g22A (A:)
    idykfwytqpvpkindefnesvnepfisdnkvedvrkdeyklppgyswyvcdvkdekdrs
    eiytlltdnyvedddnifrfnysaefllwaltspnylktwhigvkydasnkligfisaip
    tdicihkrtikmaevnflcvhktlrskrlapvlikeitrrinleniwqaiytagvylpkp
    vsdaryyhrsinvkklieigfsslnsrltmsraiklyrvedtlniknmrlmkkkdvegvh
    kllgsyleqfnlyavftkeeiahwflpienviytyvneengkikdmisfyslpsqilgnd
    kystlnaaysfynvtttatfkqlmqdaillakrnnfdvfnalevmqnksvfedlkfgegd
    gslkyylynwkcasfapahvgivll
    

  • Chain 'B':
    Sequence; same for both SEQRES and ATOM records: (download)
    >5g22B (B:)
    idykfwytqpvpkindefnesvnepfisdnkvedvrkdeyklppgyswyvcdvkdekdrs
    eiytlltdnyvedddnifrfnysaefllwaltspnylktwhigvkydasnkligfisaip
    tdicihkrtikmaevnflcvhktlrskrlapvlikeitrrinleniwqaiytagvylpkp
    vsdaryyhrsinvkklieigfsslnsrltmsraiklyrvedtlniknmrlmkkkdvegvh
    kllgsyleqfnlyavftkeeiahwflpienviytyvneengkikdmisfyslpsqilgnd
    kystlnaaysfynvtttatfkqlmqdaillakrnnfdvfnalevmqnksvfedlkfgegd
    gslkyylynwkcasfapahvgivll
    

  • Chain 'C':
    Sequence, based on SEQRES records: (download)
    >5g22C (C:)
    idykfwytqpvpkindefnesvnepfisdnkvedvrkdeyklppgyswyvcdvkdekdrs
    eiytlltdnyvedddnifrfnysaefllwaltspnylktwhigvkydasnkligfisaip
    tdicihkrtikmaevnflcvhktlrskrlapvlikeitrrinleniwqaiytagvylpkp
    vsdaryyhrsinvkklieigfsslnsrltmsraiklyrvedtlniknmrlmkkkdvegvh
    kllgsyleqfnlyavftkeeiahwflpienviytyvneengkikdmisfyslpsqilgnd
    kystlnaaysfynvtttatfkqlmqdaillakrnnfdvfnalevmqnksvfedlkfgegd
    gslkyylynwkcasfapahvgivll
    

    Sequence, based on observed residues (ATOM records): (download)
    >5g22C (C:)
    dykfwytqpvpkindefnesvnepfisdnkvedvrkdeyklppgyswyvcdvkdekdrse
    iytlltdnyvedddnifrfnysaefllwaltspnylktwhigvkydasnkligfisaipt
    dicihkrtikmaevnflcvhktlrskrlapvlikeitrrinleniwqaiytagvylpkpv
    sdaryyhrsinvkklieigfyrvedtlniknmrlmkkkdvegvhkllgsyleqfnlyavf
    tkeeiahwflpienviytyvneengkikdmisfyslpsqilgndkystlnaaysfynvtt
    tatfkqlmqdaillakrnnfdvfnalevmqnksvfedlkfgegdgslkyylynwkcasfa
    pahvgivll