PDB entry 4dhq
View 4dhq on RCSB PDB site
Description: Small-molecule inhibitors of 14-3-3 protein-protein interactions from virtual screening
Class: protein binding/inhibitor
Keywords: ADAPTER PROTEIN, PHOSPHOPROTEIN BINDING, PROTEIN BINDING-INHIBITOR complex
Deposited on
2012-01-30, released
2013-07-31
The last revision prior to the SCOPe 2.04 freeze date was dated
2013-09-04, with a file datestamp of
2013-08-30.
Experiment type: XRAY
Resolution: 1.75 Å
R-factor: 0.151
AEROSPACI score: 0.6
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 14-3-3 protein sigma
Species: Homo sapiens [TaxId:9606]
Gene: HME1, SFN
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4dhqa_ - Heterogens: MG, CL, GOL, Y06, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4dhqA (A:)
amgsmerasliqkaklaeqaeryedmaafmkgavekgeelsceernllsvayknvvggqr
aawrvlssieqksneegseekgpevreyrekvetelqgvcdtvlglldshlikeagdaes
rvfylkmkgdyyrylaevatgddkkriidsarsayqeamdiskkempptnpirlglalnf
svfhyeianspeeaislakttfdeamadlhtlsedsykdstlimqllrdnltlwt
Sequence, based on observed residues (ATOM records): (download)
>4dhqA (A:)
amgsmerasliqkaklaeqaeryedmaafmkgavekgeelsceernllsvayknvvggqr
aawrvlssieqksneekgpevreyrekvetelqgvcdtvlglldshlikeagdaesrvfy
lkmkgdyyrylaevatgddkkriidsarsayqeamdiskkempptnpirlglalnfsvfh
yeianspeeaislakttfdeamadlhtlsedsykdstlimqllrdnltlwt