PDB entry 4bdi
View 4bdi on RCSB PDB site
Description: Fragment-based screening identifies a new area for inhibitor binding to checkpoint kinase 2 (CHK2)
Class: transferase
Keywords: transferase
Deposited on
2012-10-05, released
2013-06-26
The last revision prior to the SCOPe 2.06 freeze date was dated
2013-06-26, with a file datestamp of
2013-06-21.
Experiment type: XRAY
Resolution: 2.32 Å
R-factor: 0.1896
AEROSPACI score: 0.39
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: serine/threonine-protein kinase chk2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d4bdia1, d4bdia2 - Heterogens: HAU, NO3, CL, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4bdiA (A:)
gplgshmsvypkalrdeyimsktlgsgacgevklaferktckkvaikiiskrkfaigsar
eadpalnveteieilkklnhpciikiknffdaedyyivlelmeggelfdkvvgnkrlkea
tcklyfyqmllavqylhengiihrdlkpenvllssqeedclikitdfghskilgetslmr
tlcgtptylapevlvsvgtagynravdcwslgvilficlsgyppfsehrtqvslkdqits
gkynfipevwaevsekaldlvkkllvvdpkarftteealrhpwlqdedmkrkfqdllsee
nestalpqvlaqpstsrkrpregeaegae
Sequence, based on observed residues (ATOM records): (download)
>4bdiA (A:)
msvypkalrdeyimsktlggevklaferktckkvaikiiskalnveteieilkklnhpci
ikiknffdaedyyivlelmeggelfdkvvgnkrlkeatcklyfyqmllavqylhengiih
rdlkpenvllssqeedclikitdfghskilgetslmrtlcgtptylapevlvsvgtagyn
ravdcwslgvilficlsgyppfsehrtqvslkdqitsgkynfipevwaevsekaldlvkk
llvvdpkarftteealrhpwlqdedmkrkfqdllseenestalpqvlaqp