PDB entry 4ai8
View 4ai8 on RCSB PDB site
Description: factor inhibiting hif-1 alpha in complex with daminozide
Class: oxidoreductase
Keywords: oxidoreductase, dioxygenase, metal-binding, helix-loop-helix-beta, dsbh, facial triad, transcription and epigenetic regulation, ankyrin repeat domain, beta-hydroxylation, transcription activator/inhibitor
Deposited on
2012-02-08, released
2012-10-03
The last revision prior to the SCOPe 2.04 freeze date was dated
2012-10-03, with a file datestamp of
2012-09-28.
Experiment type: XRAY
Resolution: 2.4 Å
R-factor: 0.231
AEROSPACI score: 0.3
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hypoxia-inducible factor 1-alpha inhibitor
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d4ai8a_ - Heterogens: SO4, GOL, DZA, ZN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4ai8A (A:)
gshmaataaeavasgsgepreeagalgpawdesqlrsysfptrpiprlsqsdpraeelie
neepvvltdtnlvypalkwdleylqenigngdfsvysasthkflyydekkmanfqnfkpr
snreemkfhefveklqdiqqrggeerlylqqtlndtvgrkivmdflgfnwnwinkqqgkr
gwgqltsnllligmegnvtpahydeqqnffaqikgykrcilfppdqfeclypypvhhpcd
rqsqvdfdnpdyerfpnfqnvvgyetvvgpgdvlyipmywwhhiesllnggititvnfwy
kgaptpkrieyplkahqkvaimrniekmlgealgnpqevgpllntmikgryn
Sequence, based on observed residues (ATOM records): (download)
>4ai8A (A:)
sgsgepreeagalgpawdesqlrsysfptrpiprlsqsdpraeelieneepvvltdtnlv
ypalkwdleylqenigngdfsvysasthkflyydekkmanfqnfkprsnreemkfhefve
klqdiqqrggeerlylqqtlndtvgrkivmdflgfnwnwinkqqgkrgwgqltsnlllig
megnvtpahydeqqnffaqikgykrcilfppdqfeclypypvhhpcdrqsqvdfdnpdye
rfpnfqnvvgyetvvgpgdvlyipmywwhhiesllnggititvnfwykgaptpkrieypl
kahqkvaimrniekmlgealgnpqevgpllntmikgryn