PDB entry 3lz3
View 3lz3 on RCSB PDB site
Description: Human aldose reductase mutant T113S complexed with IDD388
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: T113S mutant, TIM barrel, oxidoreductase, NADP, Phosphoprotein, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on
2010-03-01, released
2010-12-15
The last revision prior to the SCOPe 2.04 freeze date was dated
2011-08-24, with a file datestamp of
2011-08-19.
Experiment type: XRAY
Resolution: 1.03 Å
R-factor: 0.106
AEROSPACI score: 1.02
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: aldose reductase
Species: Homo sapiens [TaxId:9606]
Gene: ALR2
Database cross-references and differences (RAF-indexed):
- Uniprot P15121 (0-End)
- see remark 999 (4)
- engineered mutation (113)
Domains in SCOPe 2.04: d3lz3a_ - Heterogens: NAP, 388, BR, CIT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3lz3A (A:)
masrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahvyqnenevgvaiq
eklreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwpsgfkpgk
effpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykp
avnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaak
hnkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvca
llsctshkdypfheef
Sequence, based on observed residues (ATOM records): (download)
>3lz3A (A:)
masrillnngakmpilglgtwksppgqvteavkvaidvgyrhidcahvyqnenevgvaiq
eklreqvvkreelfivsklwctyhekglvkgacqktlsdlkldyldlylihwpsgfkpgk
effpldesgnvvpsdtnildtwaameelvdeglvkaigisnfnhlqvemilnkpglkykp
avnqiechpyltqekliqycqskgivvtaysplgspdrpwakpedpslledprikaiaak
hnkttaqvlirfpmqrnlvvipksvtperiaenfkvfdfelssqdmttllsynrnwrvca
llsctshkdypfh