PDB entry 3k3j
View 3k3j on RCSB PDB site
Description: P38alpha bound to novel DFG-out compound PF-00416121
Class: transferase
Keywords: p38alpha kinase, ATP-binding, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Serine/threonine-protein kinase, Transferase
Deposited on
2009-10-02, released
2009-11-10
The last revision prior to the SCOPe 2.07 freeze date was dated
2011-07-13, with a file datestamp of
2011-05-08.
Experiment type: XRAY
Resolution: 2 Å
R-factor: 0.196
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Homo sapiens [TaxId:9606]
Gene: MAPK14, CSBP, CSBP1, CSBP2, CSPB1, MXI2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d3k3ja_ - Heterogens: F4C, I46, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3k3jA (A:)
gsmsqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktglrvavkklsrp
fqsiihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivk
cqkltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedcelkildfglarhtdde
mtgyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrl
vgtpgaellkkissesarnyiqsltqmpkmnfanvfiganplavdllekmlvldsdkrit
aaqalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeem
es
Sequence, based on observed residues (ATOM records): (download)
>3k3jA (A:)
rptfyrqelnktiwevperyqnlspvgsggsvcaafdtktglrvavkklsrpfqsiihak
rtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnikltddhvqfl
iyqilrglkyihsadiihrdlkpsnlavnedcelkildfvatrwyrapeimlnwmhynqt
vdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesarnyiqslt
qmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpddepvadpy
dqsfesrdllidewksltydevisfvppp