PDB entry 3jvr
View 3jvr on RCSB PDB site
Description: Characterization of the Chk1 allosteric inhibitor binding site
Class: transferase
Keywords: Protein Kinase, ATP-binding, Cell cycle, Cytoplasm, DNA damage, DNA repair, Isopeptide bond, Kinase, Nucleotide-binding, Nucleus, Phosphoprotein, Polymorphism, Serine/threonine-protein kinase, Transferase, Ubl conjugation
Deposited on
2009-09-17, released
2009-10-06
The last revision prior to the SCOPe 2.04 freeze date was dated
2009-10-27, with a file datestamp of
2009-10-23.
Experiment type: XRAY
Resolution: 1.76 Å
R-factor: 0.202
AEROSPACI score: 0.51
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Serine/threonine-protein kinase Chk1
Species: Homo sapiens [TaxId:9606]
Gene: CHEK1, CHK1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.04: d3jvra_ - Heterogens: AGX, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3jvrA (A:)
avpfvedwdlvqtlgegaygevqlavnrvteeavavkivdmkravdcpenikkeicinkm
lnhenvvkfyghrregniqylfleycsggelfdriepdigmpepdaqrffhqlmagvvyl
hgigithrdikpenlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkr
refhaepvdvwscgivltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplal
lhkilvenpsaritipdikkdrwynkplkkg
Sequence, based on observed residues (ATOM records): (download)
>3jvrA (A:)
avpfvedwdlvqtlgeevqlavnrvteeavavkivdmenikkeicinkmlnhenvvkfyg
hrreiqylfleycsggelfdriepdigmpepdaqrffhqlmagvvylhgigithrdikpe
nlllderdnlkisdfglatvfrynnrerllnkmcgtlpyvapellkrrefhaepvdvwsc
givltamlagelpwdqpsdscqeysdwkekktylnpwkkidsaplallhkilvenpsari
tipdikkdrwynkplkkg