PDB entry 3ccn
View 3ccn on RCSB PDB site
Description: X-ray structure of c-Met with triazolopyridazine inhibitor.
Class: transferase
Keywords: c-Met Kinase Triazolopyridazine, ATP-binding, Glycoprotein, Membrane, Nucleotide-binding, Phosphoprotein, Proto-oncogene, Receptor, Transferase, Transmembrane, Tyrosine-protein kinase
Deposited on
2008-02-26, released
2008-04-29
The last revision prior to the SCOPe 2.06 freeze date was dated
2009-02-24, with a file datestamp of
2009-02-03.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: 0.238
AEROSPACI score: 0.43
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Hepatocyte growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: MET
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d3ccna_ - Heterogens: LKG, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>3ccnA (A:)
mqntvhidlsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlldndgkkih
cavkslnritdigevsqfltegiimkdfshpnvlsllgiclrsegsplvvlpymkhgdlr
nfirnethnptvkdligfglqvakgmkylaskkfvhrdlaarncmldekftvkvadfgla
rdmydkeyysvhnktgaklpvkwmaleslqtqkfttksdvwsfgvllwelmtrgappypd
vntfditvyllqgrrllqpeycpdplyevmlkcwhpkaemrpsfselvsrisaifstfig
ehyvhhhhhh
Sequence, based on observed residues (ATOM records): (download)
>3ccnA (A:)
lsalnpelvqavqhvvigpsslivhfnevigrghfgcvyhgtlkihcavkslnrevsqfl
tegiimkdfshpnvlsllgiclplvvlpymkhgdlrnfirnethnptvkdligfglqvak
gmkylaskkfvhrdlaarncmldekftvkvadfglardmydkeyysvhktgaklpvkwma
leslqtqkfttksdvwsfgvllwelmtrgappypdvntfditvyllqgrrllqpeycpdp
lyevmlkcwhpkaemrpsfselvsrisaifstfig