PDB entry 2xhd
View 2xhd on RCSB PDB site
Description: crystal structure of n-((2s)-5-(6-fluoro-3-pyridinyl)-2,3-dihydro-1h-inden-2-yl)-2-propanesulfonamide in complex with the ligand binding domain of the human glua2 receptor
Class: transport protein
Keywords: transport protein, ion channel
Deposited on
2010-06-14, released
2010-07-21
The last revision prior to the SCOPe 2.02 freeze date was dated
2011-06-01, with a file datestamp of
2011-05-27.
Experiment type: XRAY
Resolution: 1.8 Å
R-factor: 0.202
AEROSPACI score: 0.5
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Glutamate receptor 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot P42262 (119-262)
- PDB 2XHD (117-118)
Domains in SCOPe 2.02: d2xhda_ - Chain 'B':
Compound: Glutamate receptor 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot P42262 (119-End)
- PDB 2XHD (117-118)
Domains in SCOPe 2.02: d2xhdb_ - Heterogens: GLU, 7T9, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>2xhdA (A:)
ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
vrkskgkyayllestmneyieqrkpcdtmkvggnldskgygiatpkgsslrtpvnlavlk
lseqgvldklknkwwydkgecga
Sequence, based on observed residues (ATOM records): (download)
>2xhdA (A:)
nktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyg
ardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpie
saedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvr
kskgkyayllestmneyieqrkpcdtmkvggnldskgygiatpkgsslrtpvnlavlkls
eqgvldklknkwwydkgecga
- Chain 'B':
Sequence, based on SEQRES records: (download)
>2xhdB (B:)
ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
vrkskgkyayllestmneyieqrkpcdtmkvggnldskgygiatpkgsslrtpvnlavlk
lseqgvldklknkwwydkgecga
Sequence, based on observed residues (ATOM records): (download)
>2xhdB (B:)
ktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyga
rdadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpies
aedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvrk
skgkyayllestmneyieqrkpcdtmkvggnldskgygiatpkgsslrtpvnlavlklse
qgvldklknkwwydcg