PDB entry 6y7y
View 6y7y on RCSB PDB site
Description: Fragments KCL_771 and KCL_802 in complex with MAP kinase p38-alpha
Class: transferase
Keywords: fbdd, fragment based drug design, p38, mapk14, kinase, transferase
Deposited on
2020-03-02, released
2020-03-11
The last revision prior to the SCOPe 2.08 freeze date was dated
2020-09-30, with a file datestamp of
2020-09-25.
Experiment type: XRAY
Resolution: 1.51 Å
R-factor: N/A
AEROSPACI score: 0.56
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 14
Species: Mus musculus [TaxId:10090]
Gene: Mapk14, Crk1, Csbp1, Csbp2
Database cross-references and differences (RAF-indexed):
- Uniprot P47811
- engineered mutation (161)
Domains in SCOPe 2.08: d6y7ya_ - Heterogens: OFQ, LOT, SB4, CA, CL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>6y7yA (A:)
msqerptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktghrvavkklsrpfq
siihakrtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcq
kltddhvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfglarhtddemt
gyvatrwyrapeimlnwmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvg
tpgaellkkissesarnyiqslaqmpkmnfanvfiganplavdllekmlvldsdkritaa
qalahayfaqyhdpddepvadpydqsfesrdllidewksltydevisfvpppldqeemes
Sequence, based on observed residues (ATOM records): (download)
>6y7yA (A:)
ptfyrqelnktiwevperyqnlspvgsgaygsvcaafdtktghrvavkklsrpfqsiiha
krtyrelrllkhmkhenviglldvftparsleefndvylvthlmgadlnnivkcqkltdd
hvqfliyqilrglkyihsadiihrdlkpsnlavnedselkildfglvatrwyrapeimln
wmhynqtvdiwsvgcimaelltgrtlfpgtdhidqlklilrlvgtpgaellkkissesar
nyiqslaqmpkmnfanvfiganplavdllekmlvldsdkritaaqalahayfaqyhdpdd
epvadpydqsfesrdllidewksltydevisfvpppldqeeme