PDB entry 6q2w
View 6q2w on RCSB PDB site
Description: Crystal structure of human ROR gamma LBD in complex with a quinoline sulfonamide inverse agonist
Class: transcription
Keywords: ROR gamma, inverse agonist, nuclear hormone receptor, transcription
Deposited on
2018-12-03, released
2019-05-29
The last revision prior to the SCOPe 2.08 freeze date was dated
2019-06-12, with a file datestamp of
2019-06-07.
Experiment type: XRAY
Resolution: 1.99 Å
R-factor: N/A
AEROSPACI score: 0.32
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Nuclear receptor ROR-gamma
Species: Homo sapiens [TaxId:9606]
Gene: RORC, NR1F3, RORG, RZRG
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6q2wa_ - Chain 'B':
Compound: Nuclear receptor ROR-gamma
Species: Homo sapiens [TaxId:9606]
Gene: RORC, NR1F3, RORG, RZRG
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d6q2wb_ - Heterogens: HBW, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence; same for both SEQRES and ATOM records: (download)
>6q2wA (A:)
lteiehlvqsvcksyretcqlrledllrqrsnifsreevtgyqrksmwemwercahhlte
aiqyvvefakrlsgfmelcqndqivllkagamevvlvrmcraynadnrtvffegkyggme
lfralgcselissifdfshslsalhfsedeialytalvlinahrpglqekrkveqlqynl
elafhhhlckthrqsilaklppkgklrslcsqhverlqifq
- Chain 'B':
Sequence, based on SEQRES records: (download)
>6q2wB (B:)
lteiehlvqsvcksyretcqlrledllrqrsnifsreevtgyqrksmwemwercahhlte
aiqyvvefakrlsgfmelcqndqivllkagamevvlvrmcraynadnrtvffegkyggme
lfralgcselissifdfshslsalhfsedeialytalvlinahrpglqekrkveqlqynl
elafhhhlckthrqsilaklppkgklrslcsqhverlqifq
Sequence, based on observed residues (ATOM records): (download)
>6q2wB (B:)
lteiehlvqsvcksyretcqlrledllrqrsnifsreevtgyqrksmwemwercahhlte
aiqyvvefakrlsgfmelcqndqivllkagamevvlvrmcraynadnrtvffegkyggme
lfralgcselissifdfshslsalhfsedeialytalvlinahrpglqekrkveqlqynl
elafhhhlckthrqsilaklppkgklrslcsqhverlqif