PDB entry 6fqj

View 6fqj on RCSB PDB site
Description: GluA2(flop) G724C ligand binding core dimer bound to ZK200775 at 2.50 Angstrom resolution
Class: membrane protein
Keywords: AMPAR receptor, Ligand binding domain, Competitive antagonist, Cross-linked dimer, MEMBRANE PROTEIN
Deposited on 2018-02-14, released 2019-03-13
The last revision prior to the SCOPe 2.08 freeze date was dated 2019-10-02, with a file datestamp of 2019-09-27.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: N/A
AEROSPACI score: 0.21 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Glutamate receptor 2,Glutamate receptor 2
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Gria2, Glur2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P19491 (2-116)
      • linker (117-118)
    • Uniprot P19491 (119-End)
      • conflict (211)
    Domains in SCOPe 2.08: d6fqja_
  • Chain 'B':
    Compound: Glutamate receptor 2,Glutamate receptor 2
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Gria2, Glur2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P19491 (Start-116)
      • linker (117-118)
    • Uniprot P19491 (119-End)
      • conflict (211)
    Domains in SCOPe 2.08: d6fqjb_
  • Chain 'C':
    Compound: Glutamate receptor 2,Glutamate receptor 2
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Gria2, Glur2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P19491 (Start-116)
      • linker (117-118)
    • Uniprot P19491 (119-End)
      • conflict (211)
    Domains in SCOPe 2.08: d6fqjc_
  • Chain 'D':
    Compound: Glutamate receptor 2,Glutamate receptor 2
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Gria2, Glur2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P19491 (2-116)
      • linker (117-118)
    • Uniprot P19491 (119-End)
      • conflict (211)
    Domains in SCOPe 2.08: d6fqjd_
  • Chain 'E':
    Compound: Glutamate receptor 2,Glutamate receptor 2
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Gria2, Glur2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P19491 (Start-116)
      • linker (117-118)
    • Uniprot P19491 (119-End)
      • conflict (211)
    Domains in SCOPe 2.08: d6fqje_
  • Chain 'F':
    Compound: Glutamate receptor 2,Glutamate receptor 2
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Gria2, Glur2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P19491 (Start-116)
      • linker (117-118)
    • Uniprot P19491 (119-End)
      • conflict (211)
    Domains in SCOPe 2.08: d6fqjf_
  • Chain 'G':
    Compound: Glutamate receptor 2,Glutamate receptor 2
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Gria2, Glur2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P19491 (Start-116)
      • linker (117-118)
    • Uniprot P19491 (119-End)
      • conflict (211)
    Domains in SCOPe 2.08: d6fqjg_
  • Chain 'H':
    Compound: Glutamate receptor 2,Glutamate receptor 2
    Species: Rattus norvegicus [TaxId:10116]
    Gene: Gria2, Glur2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P19491 (Start-116)
      • linker (117-118)
    • Uniprot P19491 (119-End)
      • conflict (211)
    Domains in SCOPe 2.08: d6fqjh_
  • Heterogens: ZK1, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >6fqjA (A:)
    ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
    ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
    iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
    vrkskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlk
    lneqglldklknkwwydkgecgsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fqjA (A:)
    nktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyg
    ardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpie
    saedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvr
    kskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlkln
    eqglldklknkwwydkgecgs
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >6fqjB (B:)
    ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
    ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
    iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
    vrkskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlk
    lneqglldklknkwwydkgecgsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fqjB (B:)
    ktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyga
    rdadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpies
    aedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvrk
    skgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlklne
    qglldklknkwwydkgec
    

  • Chain 'C':
    Sequence, based on SEQRES records: (download)
    >6fqjC (C:)
    ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
    ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
    iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
    vrkskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlk
    lneqglldklknkwwydkgecgsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fqjC (C:)
    ktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyga
    rdadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpies
    aedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvrk
    skgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlklne
    qglldklknkwwydkgecg
    

  • Chain 'D':
    Sequence, based on SEQRES records: (download)
    >6fqjD (D:)
    ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
    ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
    iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
    vrkskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlk
    lneqglldklknkwwydkgecgsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fqjD (D:)
    nktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyg
    ardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpie
    saedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvr
    kskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlkln
    eqglldklknkwwydkgec
    

  • Chain 'E':
    Sequence, based on SEQRES records: (download)
    >6fqjE (E:)
    ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
    ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
    iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
    vrkskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlk
    lneqglldklknkwwydkgecgsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fqjE (E:)
    ktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyga
    rdadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpies
    aedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvrk
    skgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlklne
    qglldklknkwwydkgec
    

  • Chain 'F':
    Sequence, based on SEQRES records: (download)
    >6fqjF (F:)
    ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
    ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
    iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
    vrkskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlk
    lneqglldklknkwwydkgecgsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fqjF (F:)
    ktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyga
    rdadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpies
    aedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvrk
    skgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlklne
    qglldklknkwwydkgec
    

  • Chain 'G':
    Sequence, based on SEQRES records: (download)
    >6fqjG (G:)
    ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
    ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
    iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
    vrkskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlk
    lneqglldklknkwwydkgecgsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fqjG (G:)
    ktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyga
    rdadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpies
    aedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvrk
    skgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlklne
    qglldklknkwwydkgecgs
    

  • Chain 'H':
    Sequence, based on SEQRES records: (download)
    >6fqjH (H:)
    ganktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgk
    ygardadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtp
    iesaedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvar
    vrkskgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlk
    lneqglldklknkwwydkgecgsg
    

    Sequence, based on observed residues (ATOM records): (download)
    >6fqjH (H:)
    ktvvvttilespyvmmkknhemlegneryegycvdlaaeiakhcgfkykltivgdgkyga
    rdadtkiwngmvgelvygkadiaiapltitlvreevidfskpfmslgisimikkgtpies
    aedlskqteiaygtldsgstkeffrrskiavfdkmwtymrsaepsvfvrttaegvarvrk
    skgkyayllestmneyieqrkpcdtmkvcgnldskgygiatpkgsslgnavnlavlklne
    qglldklknkwwydkgecgs