PDB entry 5xgm
View 5xgm on RCSB PDB site
Description: Crystal structure of EGFR 696-1022 T790M in complex with Go6976
Class: transferase/transferase inhibitor
Keywords: EGFR T790M, Go6976, Inhibitor, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2017-04-14, released
2017-10-11
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-10-11, with a file datestamp of
2017-10-06.
Experiment type: XRAY
Resolution: 2.95 Å
R-factor: N/A
AEROSPACI score: 0.14
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5xgma_ - Heterogens: 85X, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5xgmA (A:)
gamggeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreat
spkankeildeayvmasvdnphvcrllgicltstvqlimqlmpfgclldyvrehkdnigs
qyllnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyha
eggkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekge
rlpqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlps
ptdsnfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>5xgmA (A:)
geapnqallrilketefkkikvlgsgagtvykglwipegekvkipvaikelrspkankei
ldeayvmasvdnphvcrllgicltstvqlimqlmpfgclldyvrehkdnigsqyllnwcv
qiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglkvpikwmalesilhriythqs
dvwsygvtvwelmtfgskpydgipaseissilekgerlpqppictidvymimvkcwmida
dsrpkfreliiefskmardpqrylviqgdermlpdmddvvdadeylip