PDB entry 5wnm
View 5wnm on RCSB PDB site
Description: Crystal structure of murine receptor-interacting protein 4 (Ripk4) D143N bound to tozasertib (VX-680)
Class: transferase/transferase inhibitor
Keywords: Kinase, Inhibitor, Complex, TRANSFERASE, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2017-08-01, released
2018-05-09
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-05-16, with a file datestamp of
2018-05-11.
Experiment type: XRAY
Resolution: 2.6 Å
R-factor: N/A
AEROSPACI score: 0.2
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Receptor-interacting serine/threonine-protein kinase 4
Species: Mus musculus [TaxId:10090]
Gene: Ripk4, Ankrd3, Pkk
Database cross-references and differences (RAF-indexed):
- Uniprot Q9ERK0
- engineered mutation (142)
Domains in SCOPe 2.08: d5wnma_ - Heterogens: CL, VX6, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5wnmA (A:)
megegrgrwalgllrtfdagefagwekvgsggfgqvykvrhvhwktwlaikcspslhvdd
rermelleeakkmemakfryilpvygicqepvglvmeymetgslekllaseplpwdlrfr
ivhetavgmnflhcmsppllhlnlkpanilldahyhvkisdfglakcngmshshdlsmdg
lfgtiaylpperireksrlfdtkhdvysfaiviwgvltqkkpfadeknilhimmkvvkgh
rpelppicrprpracasliglmqrcwhadpqvrptfqeitsetedlcekpdeevkdlahe
pgeksslesksearpessrlkrasappfdndcslsellsqld
Sequence, based on observed residues (ATOM records): (download)
>5wnmA (A:)
algllrtfdagefagwekvgsfgqvykvrhvhwktwlaikcspslhvddrermelleeak
kmemakfryilpvygicqepvglvmeymetgslekllaseplpwdlrfrivhetavgmnf
lhcmsppllhlnlkpanilldahyhvkisdfglakfgtiaylpperireksrlfdtkhdv
ysfaiviwgvltqkkpfadeknilhimmkvvkghrpelppicrprpracasliglmqrcw
hadpqvrptfqeitsetedlcek