PDB entry 5w6e

View 5w6e on RCSB PDB site
Description: PDE1b complexed with compound 3S
Class: Hydrolase/Hydrolase Inhibitor
Keywords: Phosphodiesterase, inhibitor, Hydrolase-Hydrolase Inhibitor complex
Deposited on 2017-06-16, released 2018-05-30
The last revision prior to the SCOPe 2.08 freeze date was dated 2018-06-06, with a file datestamp of 2018-06-01.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: N/A
AEROSPACI score: 0.34 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Calcium/calmodulin-dependent 3',5'-cyclic nucleotide phosphodiesterase 1B
    Species: Homo sapiens [TaxId:9606]
    Gene: PDE1B, PDE1B1, PDES1B
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d5w6ea_
  • Heterogens: ZN, MG, 0NY, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5w6eA (A:)
    gsmtytsvgptystavlnclknldlwcfdvfslnqaaddhalrtivfelltrhnlisrfk
    iptvflmsfldaletgygkyknpyhnqihaadvtqtvhcfllrtgmvhclseiellaiif
    aaaihdyehtgttnsfhiqtksecaivyndrsvlenhhissvfrlmqddemnifinltkd
    efvelralviemvlatdmschfqqvktmktalqqleridkpkalslllhaadishptkqw
    lvhsrwtkalmeeffrqgdkeaelglpfsplcdrtstlvaqsqigfidfiveptfsvltd
    vaeksvqpladedsksknqpsfqwrqpsldvevgdpnpdvvsfrstwvkriqenkqkwke
    raasgitnq
    

    Sequence, based on observed residues (ATOM records): (download)
    >5w6eA (A:)
    ystavlnclknldlwcfdvfslnqaaddhalrtivfelltrhnlisrfkiptvflmsfld
    aletgygkyknpyhnqihaadvtqtvhcfllrtgmvhclseiellaiifaaaihdyehtg
    ttnsfhiqtksecaivyndrsvlenhhissvfrlmqddemnifinltkdefvelralvie
    mvlatdmschfqqvktmktalqqleridkpkalslllhaadishptkqwlvhsrwtkalm
    eeffrqgdkeaelglpfsplcdrtstlvaqsqigfidfiveptfsvltdvaeksvqvvsf
    rstwvkriqenkqkwkeraas