PDB entry 5vnd
View 5vnd on RCSB PDB site
Description: Crystal structure of FGFR1-Y563C (FGFR4 surrogate) covalently bound to H3B-6527
Class: transferase/transferase inhibitor
Keywords: FGFR4, H3B-56527, Covalent compound, transferase-transferase inhibitor complex
Deposited on
2017-04-30, released
2017-05-24
The last revision prior to the SCOPe 2.06 freeze date was dated
2017-05-24, with a file datestamp of
2017-05-19.
Experiment type: XRAY
Resolution: 2.2 Å
R-factor: N/A
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, BFGFR, CEK, FGFBR, FLG, FLT2, HBGFR
Database cross-references and differences (RAF-indexed):
- Uniprot P11362 (Start-308)
- engineered mutation (31)
- engineered mutation (106)
- engineered mutation (127)
Domains in SCOPe 2.06: d5vnda_ - Chain 'B':
Compound: fibroblast growth factor receptor 1
Species: Homo sapiens [TaxId:9606]
Gene: FGFR1, BFGFR, CEK, FGFBR, FLG, FLT2, HBGFR
Database cross-references and differences (RAF-indexed):
- Uniprot P11362 (Start-308)
- engineered mutation (31)
- engineered mutation (106)
Domains in SCOPe 2.06: d5vndb_ - Heterogens: 9ES, SO4, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5vndA (A:)
gagvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkml
ksdatekdlsdlisememmkmigkhkniinllgactqdgplyvivecaskgnlreylqar
rppgleysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednv
mkiadfglardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftl
ggspypgvpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldr
ivaltsnqe
Sequence, based on observed residues (ATOM records): (download)
>5vndA (A:)
yelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkmlksdate
kdlsdlisememmkmigkhkniinllgactqdgplyvivecaskgnlreylqarrppgle
ysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadf
glardhhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypg
vpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivaltsn
qe
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5vndB (B:)
gagvseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkml
ksdatekdlsdlisememmkmigkhkniinllgactqdgplyvivecaskgnlreylqar
rppgleysynpshnpeeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednv
mkiadfglardihhidyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftl
ggspypgvpveelfkllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldr
ivaltsnqe
Sequence, based on observed residues (ATOM records): (download)
>5vndB (B:)
vseyelpedprwelprdrlvlgkplgegafgqvvlaeaigldkdkpnrvtkvavkmlksd
atekdlsdlisememmkmigkhkniinllgactqdgplyvivecaskgnlreylqarrpp
geeqlsskdlvscayqvargmeylaskkcihrdlaarnvlvtednvmkiadfglardihh
idyykkttngrlpvkwmapealfdriythqsdvwsfgvllweiftlggspypgvpveelf
kllkeghrmdkpsnctnelymmmrdcwhavpsqrptfkqlvedldrivaltsnqe