PDB entry 5u43
View 5u43 on RCSB PDB site
Description: Human PPARdelta ligand-binding domain in complexed with specific agonist 12
Class: protein binding/activator
Keywords: PPARdelta, ligand-binding domain, agonist, PROTEIN BINDING-ACTIVATOR complex
Deposited on
2016-12-03, released
2017-03-22
The last revision prior to the SCOPe 2.08 freeze date was dated
2020-07-29, with a file datestamp of
2020-07-04.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: N/A
AEROSPACI score: 0.45
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Peroxisome proliferator-activated receptor delta
Species: Homo sapiens [TaxId:9606]
Gene: PPARD, NR1C2, PPARB
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5u43a_ - Chain 'B':
Compound: Peroxisome proliferator-activated receptor delta
Species: Homo sapiens [TaxId:9606]
Gene: PPARD, NR1C2, PPARB
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5u43b_ - Heterogens: 7SS, PGO, PEG, B7G, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5u43A (A:)
pqvadlkafskhiynaylknfnmtkkkarsiltgkashtapfvihdietlwqaekglvwk
qlvnglppykeisvhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygvhea
ifamlasivnkdgllvangsgfvtreflrslrkpfsdiiepkfefavkfnalelddsdla
lfiaaiilcgdrpglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadlrql
vtehaqmmqrikktetetslhpllqeiykdmy
Sequence, based on observed residues (ATOM records): (download)
>5u43A (A:)
pqvadlkafskhiynaylknfnmtkkkarsiltgkapfvihdietlwqaekglvwkqlvn
glppykeisvhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygvheaifam
lasivnkdgllvangsgfvtreflrslrkpfsdiiepkfefavkfnalelddsdlalfia
aiilcgdrpglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadlrqlvteh
aqmmqrikktetetslhpllqeiykd
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5u43B (B:)
pqvadlkafskhiynaylknfnmtkkkarsiltgkashtapfvihdietlwqaekglvwk
qlvnglppykeisvhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygvhea
ifamlasivnkdgllvangsgfvtreflrslrkpfsdiiepkfefavkfnalelddsdla
lfiaaiilcgdrpglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadlrql
vtehaqmmqrikktetetslhpllqeiykdmy
Sequence, based on observed residues (ATOM records): (download)
>5u43B (B:)
dlkafskhiynaylknfnmtkkkarsiltgapfvihdietlwqaekglvwkqlvnglppy
keisvhvfyrcqcttvetvreltefaksipsfsslflndqvtllkygvheaifamlasiv
nkdgllvangsgfvtreflrslrkpfsdiiepkfefavkfnalelddsdlalfiaaiilc
gdrpglmnvprveaiqdtilralefhlqanhpdaqylfpkllqkmadlrqlvtehaqmmq
rikktetetslhpllqeiykdm