PDB entry 5qik
View 5qik on RCSB PDB site
Description: TGF-BETA RECEPTOR TYPE 1 KINASE DOMAIN (T204D) IN COMPLEX WITH N-{4-[3-(6-fluoropyridin-3-yl)-4-oxo-4,5,6,7-tetrahydro-1H-pyrrolo[3,2-c]pyridin-2-yl]pyridin-2-yl}acetamide
Class: transferase/transferase inhibitor
Keywords: alk5, sb431542, kinase domain, transferase-transferase inhibitor complex, transferase
Deposited on
2018-08-05, released
2018-10-31
The last revision prior to the SCOPe 2.08 freeze date was dated
2021-05-12, with a file datestamp of
2021-05-07.
Experiment type: XRAY
Resolution: 1.58 Å
R-factor: N/A
AEROSPACI score: 0.54
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: TGF-beta receptor type-1
Species: Homo sapiens [TaxId:9606]
Gene: TGFBR1, ALK5, SKR4
Database cross-references and differences (RAF-indexed):
- Uniprot P36897 (3-End)
- expression tag (0-2)
- engineered mutation (7)
Domains in SCOPe 2.08: d5qika1, d5qika2 - Heterogens: J2M, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5qikA (A:)
ghmtiardivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrh
enilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahl
hmeivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtk
rymapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdp
sveemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqls
qqegikm
Sequence, based on observed residues (ATOM records): (download)
>5qikA (A:)
ghmtiardivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrh
enilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahl
hmeivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtk
rymapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdp
sveemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqls
qqe