PDB entry 5nhh

View 5nhh on RCSB PDB site
Description: Human Erk2 with an Erk1/2 inhibitor
Class: transferase
Keywords: Erk2, kinase, inhibitor, oncology, TRANSFERASE
Deposited on 2017-03-21, released 2017-04-19
The last revision prior to the SCOPe 2.08 freeze date was dated 2017-05-10, with a file datestamp of 2017-05-05.
Experiment type: XRAY
Resolution: 1.94 Å
R-factor: N/A
AEROSPACI score: 0.33 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: Mitogen-activated protein kinase 1
    Species: Homo sapiens [TaxId:9606]
    Gene: MAPK1, ERK2, PRKM1, PRKM2
    Database cross-references and differences (RAF-indexed):
    • Uniprot P28482
      • conflict (64)
    Domains in SCOPe 2.08: d5nhha_
  • Heterogens: SO4, 8XH, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5nhhA (A:)
    mhhhhhhgggenlyfqgshmaaaaaagagpemvrgqvfdvgprytnlsyigegaygmvcs
    aydnlnkvrvaikkispfehqtycqrtlreikillrfrheniigindiiraptieqmkdv
    yivqdlmetdlykllktqhlsndhicyflyqilrglkyihsanvlhrdlkpsnlllnttc
    dlkicdfglarvadpdhdhtgflteyvatrwyrapeimlnskgytksidiwsvgcilaem
    lsnrpifpgkhyldqlnhilgilgspsqedlnciinlkarnyllslphknkvpwnrlfpn
    adskaldlldkmltfnphkrieveqalahpyleqyydpsdepiaeapfkfdmelddlpke
    klkelifeetarfqpgyrsle
    

    Sequence, based on observed residues (ATOM records): (download)
    >5nhhA (A:)
    pemvrgqvfdvgprytnlsyigegaygmvcsaydnlnkvrvaikkispfehqtycqrtlr
    eikillrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyfl
    yqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadpdhdhtgflteyvat
    rwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsqe
    dlnciinlkarnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqalah
    pyleqyydpsdepiaeapfkfdmelddlpkeklkelifeetarfqpgy