PDB entry 5mzg
View 5mzg on RCSB PDB site
Description: Crystal structure of mouse MTH1 in complex with TH588
Class: hydrolase
Keywords: Inhibitor, complex, hydrolase
Deposited on
2017-01-31, released
2018-01-10
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-02-14, with a file datestamp of
2018-02-09.
Experiment type: XRAY
Resolution: 1.85 Å
R-factor: N/A
AEROSPACI score: 0.36
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 7,8-dihydro-8-oxoguanine triphosphatase
Species: Mus musculus [TaxId:10090]
Gene: NUDT1, MTH1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5mzga1, d5mzga2 - Chain 'B':
Compound: 7,8-dihydro-8-oxoguanine triphosphatase
Species: Mus musculus [TaxId:10090]
Gene: NUDT1, MTH1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5mzgb_ - Heterogens: 2GE, SO4, SCN, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5mzgA (A:)
mgsshhhhhhssglvprgshmstsrlytlvlvlqpqrvllgmkkrgfgagrwngfggkvq
egetiedgakrelleesglsvdtlhkvghisfefvgspelmdvhifsadhvhgtptesee
mrpqwfqldqipfadlwpddsywfplllqkkkfcghfkfqdqdtilsyslrevdsf
Sequence, based on observed residues (ATOM records): (download)
>5mzgA (A:)
hmstsrlytlvlvlqpqrvllgmkkrgfgagrwngfggkvqegetiedgakrelleesgl
svdtlhkvghisfefvgspelmdvhifsadhvhgtpteseemrpqwfqldqipfadlwpd
dsywfplllqkkkfcghfkfqdqdtilsyslrevd
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5mzgB (B:)
mgsshhhhhhssglvprgshmstsrlytlvlvlqpqrvllgmkkrgfgagrwngfggkvq
egetiedgakrelleesglsvdtlhkvghisfefvgspelmdvhifsadhvhgtptesee
mrpqwfqldqipfadlwpddsywfplllqkkkfcghfkfqdqdtilsyslrevdsf
Sequence, based on observed residues (ATOM records): (download)
>5mzgB (B:)
mstsrlytlvlvlqpqrvllgmkkrgfgagrwngfggkvqegetiedgakrelleesgls
vdtlhkvghisfefvgspelmdvhifsadhvhgtpteseemrpqwfqldqipfadlwpdd
sywfplllqkkkfcghfkfqdqdtilsyslrev