PDB entry 5mfw
View 5mfw on RCSB PDB site
Description: Crystal structure of the GluK1 ligand-binding domain in complex with kainate and BPAM-121 at 2.10 A resolution
Class: membrane protein
Keywords: ionotropic glutamate receptor, GluK1 ligand-binding domain, membrane protein, positive allosteric modulator
Deposited on
2016-11-18, released
2017-04-12
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-01-17, with a file datestamp of
2018-01-12.
Experiment type: XRAY
Resolution: 2.1 Å
R-factor: N/A
AEROSPACI score: 0.29
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Grik1, Glur5
Database cross-references and differences (RAF-indexed):
- Uniprot P22756 (Start-115)
- see remark 999 (33)
- linker (116-117)
- Uniprot P22756 (118-End)
Domains in SCOPe 2.08: d5mfwa_ - Chain 'B':
Compound: Glutamate receptor ionotropic, kainate 1,Glutamate receptor ionotropic, kainate 1
Species: Rattus norvegicus [TaxId:10116]
Gene: Grik1, Glur5
Database cross-references and differences (RAF-indexed):
- Uniprot P22756 (Start-115)
- see remark 999 (33)
- linker (116-117)
- Uniprot P22756 (118-256)
Domains in SCOPe 2.08: d5mfwb_ - Heterogens: 7M6, CL, KAI, SO4, GOL, ACT, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5mfwA (A:)
ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
gklhmmkekwwrgngcp
Sequence, based on observed residues (ATOM records): (download)
>5mfwA (A:)
nrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkyg
aqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpids
addlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvlt
tdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegk
lhmmkekww
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5mfwB (B:)
ganrtlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgk
ygaqndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpi
dsaddlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrv
lttdyallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqee
gklhmmkekwwrgngcp
Sequence, based on observed residues (ATOM records): (download)
>5mfwB (B:)
tlivttileepyvmyrksdkplygndrfegycldllkelsnilgflydvklvpdgkygaq
ndkgewngmvkelidhradlavapltityvrekvidfskpfmtlgisilyrkgtpidsad
dlakqtkieygavrdgstmtffkkskistyekmwafmssrqqsalvknsdegiqrvlttd
yallmestsieyvtqrncnltqigglidskgygvgtpigspyrdkitiailqlqeegklh
mmkekwwrgngcp