PDB entry 5mae
View 5mae on RCSB PDB site
Description: CATHEPSIN L IN COMPLEX WITH (2S,4R)-4-(2-Chloro-4-methoxy-benzenesulfonyl)-1-[3-(5-chloro-pyridin-2-yl)-azetidine-3-carbonyl]-pyrrolidine-2-car boxylic acid (1-cyano-cyclopropyl)-amide
Class: hydrolase
Keywords: protease inhibitor, hydrolase-hydrolase inhibitor complex, hydrolase
Deposited on
2016-11-03, released
2017-01-11
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-02-22, with a file datestamp of
2017-02-17.
Experiment type: XRAY
Resolution: 1 Å
R-factor: N/A
AEROSPACI score: 0.81
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Cathepsin L1
Species: Homo sapiens [TaxId:9606]
Gene: CTSL, CTSL1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5maea_ - Heterogens: 7KN, EDO, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5maeA (A:)
aprsvdwrekgyvtpvknqgqcgscwafsatgalegqmfrktgrlislseqnlvdcsgpq
gnegcngglmdyafqyvqdnggldseesypyeateesckynpkysvandtgfvdipkqek
almkavatvgpisvaidaghesflfykegiyfepdcssedmdhgvlvvgygfestesdnn
kywlvknswgeewgmggyvkmakdrrnhcgiasaasyptv
Sequence, based on observed residues (ATOM records): (download)
>5maeA (A:)
aprsvdwrekgyvtpvknqgqcgscwafsatgalegqmfrktgrlislseqnlvdcsgpq
gnegcngglmdyafqyvqdnggldseesypyeateesckynpkysvandtgfvdipkqek
almkavatvgpisvaidaghesflfykegiyfepdcssedmdhgvlvvgygfestnnkyw
lvknswgeewgmggyvkmakdrrnhcgiasaasyptv