PDB entry 5lcj
View 5lcj on RCSB PDB site
Description: In-Gel Activity-Based Protein Profiling of a Clickable Covalent Erk 1/2 Inhibitor
Class: transferase
Keywords: Erk1/2 covalent inhibitor, TRANSFERASE
Deposited on
2016-06-22, released
2016-07-20
The last revision prior to the SCOPe 2.08 freeze date was dated
2016-08-31, with a file datestamp of
2016-08-24.
Experiment type: XRAY
Resolution: 1.78 Å
R-factor: N/A
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Mitogen-activated protein kinase 1
Species: Homo sapiens [TaxId:9606]
Gene: MAPK1, ERK2, PRKM1, PRKM2
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5lcja_ - Heterogens: 6TS, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5lcjA (A:)
mahhhhhhmaaaaaagagpemvrgqvfdvgprytnlsyigegaygmvcsaydnvnkvrva
ikkispfehqtycqrtlreikillrfrheniigindiiraptieqmkdvyivqdlmetdl
ykllktqhlsndhicyflyqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglar
vadpdhdhtgflteyvatrwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkh
yldqlnhilgilgspsqedlnciinlkarnyllslphknkvpwnrlfpnadskaldlldk
mltfnphkrieveqalahpyleqyydpsdepiaeapfkfdmelddlpkeklkelifeeta
rfqpgyrs
Sequence, based on observed residues (ATOM records): (download)
>5lcjA (A:)
pemvrgqvfdvgprytnlsyigegaygmvcsaydnvnkvrvaikkispfehqtycqrtlr
eikillrfrheniigindiiraptieqmkdvyivqdlmetdlykllktqhlsndhicyfl
yqilrglkyihsanvlhrdlkpsnlllnttcdlkicdfglarvadpdhdhtgflteyvat
rwyrapeimlnskgytksidiwsvgcilaemlsnrpifpgkhyldqlnhilgilgspsqe
dlnciinlkarnyllslphknkvpwnrlfpnadskaldlldkmltfnphkrieveqalah
pyleqyydpsdepiaeapfkfdelddlpkeklkelifeetarfqpg