PDB entry 5kad
View 5kad on RCSB PDB site
Description: Protein Tyrosine Phosphatase 1B N193A mutant in complex with TCS401, closed state
Class: hydrolase/hydrolase inhibitor
Keywords: Protein tyrosine phosphatase, hydrolase-hydrolase inhibitor complex
Deposited on
2016-06-01, released
2017-03-01
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-03-01, with a file datestamp of
2017-02-24.
Experiment type: XRAY
Resolution: 1.9 Å
R-factor: N/A
AEROSPACI score: 0.34
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: tyrosine-protein phosphatase non-receptor type 1
Species: Homo sapiens [TaxId:9606]
Gene: PTPN1, PTP1B
Database cross-references and differences (RAF-indexed):
- Uniprot P18031 (5-End)
- expression tag (1-4)
- engineered mutation (197)
Domains in SCOPe 2.08: d5kada1, d5kada2 - Chain 'B':
Compound: tyrosine-protein phosphatase non-receptor type 1
Species: Homo sapiens [TaxId:9606]
Gene: PTPN1, PTP1B
Database cross-references and differences (RAF-indexed):
- Uniprot P18031 (5-End)
- expression tag (2-4)
- engineered mutation (197)
Domains in SCOPe 2.08: d5kadb1, d5kadb2 - Heterogens: OTA, CL, TRS, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5kadA (A:)
ghmasmemekefeqidksgswaaiyqdirheasdfpcrvaklpknknrnryrdvspfdhs
riklhqedndyinaslikmeeaqrsyiltqgplpntcghfwemvweqksrgvvmlnrvme
kgslkcaqywpqkeekemifedtnlkltlisediksyytvrqlelenlttqetreilhfh
yttwpdfgvpespasflaflfkvresgslspehgpvvvhcsagigrsgtfcladtclllm
dkrkdpssvdikkvllemrkfrmgliqtadqlrfsylaviegakfimgdssvqdqwkels
hedlep
Sequence, based on observed residues (ATOM records): (download)
>5kadA (A:)
hmasmemekefeqidksgswaaiyqdirheasdfpcrvaklpknknrnryrdvspfdhsr
iklhqedndyinaslikmeeaqrsyiltqgplpntcghfwemvweqksrgvvmlnrvmek
gslkcaqywpqkeekemifedtnlkltlisediksyytvrqlelenlttqetreilhfhy
ttwpdfgvpespasflaflfkvresgslspehgpvvvhcsagigrsgtfcladtclllmd
krkdpssvdikkvllemrkfrmgliqtadqlrfsylaviegakfi
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5kadB (B:)
ghmasmemekefeqidksgswaaiyqdirheasdfpcrvaklpknknrnryrdvspfdhs
riklhqedndyinaslikmeeaqrsyiltqgplpntcghfwemvweqksrgvvmlnrvme
kgslkcaqywpqkeekemifedtnlkltlisediksyytvrqlelenlttqetreilhfh
yttwpdfgvpespasflaflfkvresgslspehgpvvvhcsagigrsgtfcladtclllm
dkrkdpssvdikkvllemrkfrmgliqtadqlrfsylaviegakfimgdssvqdqwkels
hedlep
Sequence, based on observed residues (ATOM records): (download)
>5kadB (B:)
masmemekefeqidksgswaaiyqdirheasdfpcrvaklpknknrnryrdvspfdhsri
klhqedndyinaslikmeeaqrsyiltqgplpntcghfwemvweqksrgvvmlnrvmekg
slkcaqywpqkeekemifedtnlkltlisediksyytvrqlelenlttqetreilhfhyt
twpdfgvpespasflaflfkvresgslspehgpvvvhcsagigrsgtfcladtclllmdk
rksvdikkvllemrkfrmgliqtadqlrfsylaviegakfim