PDB entry 5jv2
View 5jv2 on RCSB PDB site
Description: Crystal structure of human FPPS in complex with an allosteric inhibitor MIT-01-055
Class: transferase/transferase inhibitor
Keywords: Transferase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2016-05-10, released
2017-03-15
The last revision prior to the SCOPe 2.08 freeze date was dated
2017-03-22, with a file datestamp of
2017-03-17.
Experiment type: XRAY
Resolution: 2.3 Å
R-factor: N/A
AEROSPACI score: 0.25
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'F':
Compound: farnesyl pyrophosphate synthase
Species: Homo sapiens [TaxId:9606]
Gene: FDPS, FPS, KIAA1293
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5jv2f_ - Heterogens: PO4, CL, 6O3, HOH
PDB Chain Sequences:
- Chain 'F':
Sequence, based on SEQRES records: (download)
>5jv2F (F:)
mgsshhhhhhssgrenlyfqghmngdqnsdvyaqekqdfvqhfsqivrvltedemghpei
gdaiarlkevleynaiggkynrgltvvvafrelveprkqdadslqrawtvgwcvellqaf
flvaddimdssltrrgqicwyqkpgvgldaindanlleaciyrllklycreqpyylnlie
lflqssyqteigqtldlltapqgnvdlvrftekryksivkyktafysfylpiaaamymag
idgekehanakkillemgeffqiqddyldlfgdpsvtgkigtdiqdnkcswlvvqclqra
tpeqyqilkenygqkeaekvarvkalyeeldlpavflqyeedsyshimalieqyaaplpp
avflglarkiykrrk
Sequence, based on observed residues (ATOM records): (download)
>5jv2F (F:)
yaqekqdfvqhfsqivrvltepeigdaiarlkevleynaiggkynrgltvvvafrelvpr
kqdadslqrawtvgwcvellqafflvaddimdssltrrgqicwyqkpgvgldaindanll
eaciyrllklycreqpyylnlielflqssyqteigqtldlltapqgnvdlvrftekryks
ivkyktafysfylpiaaamymagidgekehanakkillemgeffqiqddyldlfgdpkig
tdiqdnkcswlvvqclqratpeqyqilkenygqkeaekvarvkalyeeldlpavflqyee
dsyshimalieqyaaplppavflglarkiyk