PDB entry 5fzj
View 5fzj on RCSB PDB site
Description: Structure of the Keap1 Kelch domain in complex with a small molecule inhibitor.
Class: transcription
Keywords: transcription, keap1, nrf2, oxidative stress
Deposited on
2016-03-14, released
2016-04-13
The last revision prior to the SCOPe 2.08 freeze date was dated
2018-04-04, with a file datestamp of
2018-03-29.
Experiment type: XRAY
Resolution: 2.01 Å
R-factor: N/A
AEROSPACI score: 0.31
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Kelch-like ECH-associated protein 1
Species: Mus musculus [TaxId:10090]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5fzja_ - Heterogens: 75K, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5fzjA (A:)
gpkvgrliytaggyfrqslsyleaynpsngswlrladlqvprsglagcvvggllyavggr
nnspdgntdssaldcynpmtnqwspcasmsvprnrigvgvidghiyavggshgcihhssv
eryeperdewhlvapmltrrigvgvavlnrllyavggfdgtnrlnsaecyypernewrmi
tpmntirsgagvcvlhnciyaaggydgqdqlnsverydvetetwtfvapmrhhrsalgit
vhqgkiyvlggydghtfldsvecydpdsdtwsevtrmtsgrsgvgvavtmepcrkqidqq
nctc
Sequence, based on observed residues (ATOM records): (download)
>5fzjA (A:)
grliytaggyfrqslsyleaynpsngswlrladlqvprsglagcvvggllyavggrnnsp
dgntdssaldcynpmtnqwspcasmsvprnrigvgvidghiyavggshgcihhssverye
perdewhlvapmltrrigvgvavlnrllyavggfdgtnrlnsaecyypernewrmitpmn
tirsgagvcvlhnciyaaggydgqdqlnsverydvetetwtfvapmrhhrsalgitvhqg
kiyvlggydghtfldsvecydpdsdtwsevtrmtsgrsgvgvavtmepc