PDB entry 5fqv
View 5fqv on RCSB PDB site
Description: Selective estrogen receptor downregulator antagonists: Tetrahydroisoquinoline phenols 5.
Class: signaling protein
Keywords: signaling protein, breast cancer, estrogen receptor downregulator, fulvestrant, thiq, nuclear hormone receptor
Deposited on
2015-12-14, released
2016-02-10
The last revision prior to the SCOPe 2.06 freeze date was dated
2016-02-10, with a file datestamp of
2016-02-05.
Experiment type: XRAY
Resolution: 1.74 Å
R-factor: N/A
AEROSPACI score: 0.4
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Estrogen receptor alpha
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
- Uniprot P03372 (0-End)
- engineered mutation (74)
- engineered mutation (110)
- engineered mutation (229)
Domains in SCOPe 2.06: d5fqva_ - Heterogens: VQI, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5fqvA (A:)
alsltadqmvsalldaeppilyseydptrpfseasmmglltnladrelvhminwakrvpg
fvdltlhdqvhllesawleilmiglvwrsmehpgkllfapnllldrnqgksvegmveifd
mllatssrfrmmnlqgeefvclksiillnsgvytflsstlksleekdhihrvldkitdtl
ihlmakagltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvpsydlllemlda
hrlhapts
Sequence, based on observed residues (ATOM records): (download)
>5fqvA (A:)
alsltadqmvsalldaeppilyseydptrpfsmmglltnladrelvhminwakrvpgfvd
ltlhdqvhllesawleilmiglvwrsmehpgkllfapnllldrnqgksvegmveifdmll
atssrfrmmnlqgeefvclksiillnsgvytftlksleekdhihrvldkitdtlihlmak
agltlqqqhqrlaqlllilshirhmsnkgmehlysmkcknvvpsydlllemld