PDB entry 5fed
View 5fed on RCSB PDB site
Description: EGFR kinase domain in complex with a covalent aminobenzimidazole inhibitor.
Class: transferase/transferase inhibitor
Keywords: Kinase, Inhibitor, Covalently-bound, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2015-12-16, released
2016-07-27
The last revision prior to the SCOPe 2.08 freeze date was dated
2016-08-10, with a file datestamp of
2016-08-05.
Experiment type: XRAY
Resolution: 2.65 Å
R-factor: N/A
AEROSPACI score: 0.19
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5feda_ - Heterogens: 5X4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5fedA (A:)
ggeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreatspk
ankeildeayvmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqyl
lnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfglakllgaeekeyhaegg
kvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerlp
qppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpsptd
snfyralmdeedmddvvdadeylipqqg
Sequence, based on observed residues (ATOM records): (download)
>5fedA (A:)
eapnqallrilketefkkikvlgsgtvykglwipegekvkipvaikespkankeildeay
vmasvdnphvcrllgicltstvqlitqlmpfgclldyvrehkdnigsqyllnwcvqiakg
mnyledrrlvhrdlaarnvlvktpqhvkitdfglakllkeyhaeggkvpikwmalesilh
riythqsdvwsygvtvwelmtfgskpydgipaseissilekgerlpqppictidvymimv
kcwmidadsrpkfreliiefskmardpqrylviqgdemddvvdadeyl