PDB entry 5f25
View 5f25 on RCSB PDB site
Description: Crystal structure of the BRD9 bromodomain in complex with compound 4.
Class: transcription
Keywords: Bromodomain, Inhibitor, transcription
Deposited on
2015-12-01, released
2016-03-09
The last revision prior to the SCOPe 2.07 freeze date was dated
2016-06-08, with a file datestamp of
2016-06-03.
Experiment type: XRAY
Resolution: 1.68 Å
R-factor: N/A
AEROSPACI score: 0.42
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: brd9
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d5f25a_ - Chain 'B':
Compound: brd9
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.07: d5f25b_ - Heterogens: 5TU, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5f25A (A:)
smlklsaenestpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmk
dkivaneyksvtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkr
sms
Sequence, based on observed residues (ATOM records): (download)
>5f25A (A:)
stpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmkdkivaneyks
vtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkrsms
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5f25B (B:)
smlklsaenestpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmk
dkivaneyksvtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkr
sms
Sequence, based on observed residues (ATOM records): (download)
>5f25B (B:)
estpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmkdkivaneyk
svtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkrsm