PDB entry 5f25

View 5f25 on RCSB PDB site
Description: Crystal structure of the BRD9 bromodomain in complex with compound 4.
Class: transcription
Keywords: Bromodomain, Inhibitor, transcription
Deposited on 2015-12-01, released 2016-03-09
The last revision prior to the SCOPe 2.07 freeze date was dated 2016-06-08, with a file datestamp of 2016-06-03.
Experiment type: XRAY
Resolution: 1.68 Å
R-factor: N/A
AEROSPACI score: 0.42 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: brd9
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d5f25a_
  • Chain 'B':
    Compound: brd9
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.07: d5f25b_
  • Heterogens: 5TU, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >5f25A (A:)
    smlklsaenestpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmk
    dkivaneyksvtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkr
    sms
    

    Sequence, based on observed residues (ATOM records): (download)
    >5f25A (A:)
    stpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmkdkivaneyks
    vtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkrsms
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >5f25B (B:)
    smlklsaenestpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmk
    dkivaneyksvtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkr
    sms
    

    Sequence, based on observed residues (ATOM records): (download)
    >5f25B (B:)
    estpiqqllehflrqlqrkdphgffafpvtdaiapgysmiikhpmdfgtmkdkivaneyk
    svtefkadfklmcdnamtynrpdtvyyklakkilhagfkmmskerllalkrsm