PDB entry 5ezv
View 5ezv on RCSB PDB site
Description: X-ray crystal structure of AMP-activated protein kinase alpha-2/alpha-1 RIM chimaera (alpha-2(1-347)/alpha-1(349-401)/alpha-2(397-end) beta-1 gamma-1) co-crystallized with C2 (5-(5-hydroxyl-isoxazol-3-yl)-furan-2-phosphonic acid)
Class: transferase
Keywords: Transferase, serine/threonine kinase, allosteric activation, nucleotide-binding
Deposited on
2015-11-26, released
2016-03-09
The last revision prior to the SCOPe 2.06 freeze date was dated
2016-03-23, with a file datestamp of
2016-03-18.
Experiment type: XRAY
Resolution: 2.99 Å
R-factor: N/A
AEROSPACI score: 0.14
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 5'-AMP-activated protein kinase catalytic subunit alpha-2/alpha-1 RIM SWAP chimera
Species: Homo sapiens [TaxId:9606]
Gene: PRKAA2, AMPK, AMPK2
Database cross-references and differences (RAF-indexed):
- Chain 'B':
Compound: 5'-AMP-activated protein kinase subunit beta-1
Species: Homo sapiens [TaxId:9606]
Gene: PRKAB1, AMPK
Database cross-references and differences (RAF-indexed):
- Chain 'C':
Compound: 5'-AMP-activated protein kinase catalytic subunit alpha-2/alpha-1 RIM SWAP chimera
Species: Homo sapiens [TaxId:9606]
Gene: PRKAA2, AMPK, AMPK2
Database cross-references and differences (RAF-indexed):
- Chain 'D':
Compound: 5'-AMP-activated protein kinase subunit beta-1
Species: Homo sapiens [TaxId:9606]
Gene: PRKAB1, AMPK
Database cross-references and differences (RAF-indexed):
- Chain 'E':
Compound: 5'-amp-activated protein kinase subunit gamma-1
Species: Homo sapiens [TaxId:9606]
Gene: Prkag1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d5ezve1, d5ezve2 - Chain 'F':
Compound: 5'-amp-activated protein kinase subunit gamma-1
Species: Homo sapiens [TaxId:9606]
Gene: Prkag1
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.06: d5ezvf1, d5ezvf2 - Heterogens: STU, C1V, C2Z, HOH
PDB Chain Sequences:
- Chain 'A':
No sequence available.
- Chain 'B':
No sequence available.
- Chain 'C':
No sequence available.
- Chain 'D':
No sequence available.
- Chain 'E':
Sequence, based on SEQRES records: (download)
>5ezvE (E:)
madlnwetvissdsspavenehpqetpesnnsvytsfmkshrcydliptssklvvfdtsl
qvkkaffalvtngvraaplwdskkqsfvgmltitdfinilhryyksalvqiyeleehkie
twrevylqdsfkplvcispnaslfdavsslirnkihrlpvidpesgntlyilthkrilkf
lklfitefpkpefmsksleelqigtyaniamvrtttpvyvalgifvqhrvsalpvvdekg
rvvdiyskfdvinlaaektynnldvsvtkalqhrshyfegvlkcylhetletiinrlvea
evhrlvvvdendvvkgivslsdilqalvltggekkp
Sequence, based on observed residues (ATOM records): (download)
>5ezvE (E:)
snnsvytsfmkshrcydliptssklvvfdtslqvkkaffalvtngvraaplwdskkqsfv
gmltitdfinilhryyksalvqiyeleehkietwrevylqsfkplvcispnaslfdavss
lirnkihrlpvidpesgntlyilthkrilkflklfitefpkpefmsksleelqigtyani
amvrtttpvyvalgifvqhrvsalpvvdekgrvvdiyskfdvinlaaektynnldvsvtk
alqhrshyfegvlkcylhetletiinrlveaevhrlvvvdendvvkgivslsdilqalvl
tg
- Chain 'F':
Sequence, based on SEQRES records: (download)
>5ezvF (F:)
madlnwetvissdsspavenehpqetpesnnsvytsfmkshrcydliptssklvvfdtsl
qvkkaffalvtngvraaplwdskkqsfvgmltitdfinilhryyksalvqiyeleehkie
twrevylqdsfkplvcispnaslfdavsslirnkihrlpvidpesgntlyilthkrilkf
lklfitefpkpefmsksleelqigtyaniamvrtttpvyvalgifvqhrvsalpvvdekg
rvvdiyskfdvinlaaektynnldvsvtkalqhrshyfegvlkcylhetletiinrlvea
evhrlvvvdendvvkgivslsdilqalvltggekkp
Sequence, based on observed residues (ATOM records): (download)
>5ezvF (F:)
nnsvytsfmkshrcydliptssklvvfdtslqvkkaffalvtngvraaplwdskkqsfvg
mltitdfinilhryyksalvqiyeleehkietwrevylqdsfkplvcispnaslfdavss
lirnkihrlpvidpesgntlyilthkrilkflklfitefpkpefmsksleelqigtyani
amvrtttpvyvalgifvqhrvsalpvvdekgrvvdiyskfdvinlaaektynnldvsvtk
alqhrshyfegvlkcylhetletiinrlveaevhrlvvvdendvvkgivslsdilqalvl