PDB entry 5edp
View 5edp on RCSB PDB site
Description: EGFR kinase (T790M/L858R) apo
Class: transferase/transferase inhibitor
Keywords: protein kinase, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2015-10-21, released
2015-12-02
The last revision prior to the SCOPe 2.08 freeze date was dated
2016-01-20, with a file datestamp of
2016-01-15.
Experiment type: XRAY
Resolution: 2.9 Å
R-factor: N/A
AEROSPACI score: 0.15
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Epidermal growth factor receptor
Species: Homo sapiens [TaxId:9606]
Gene: EGFR, ERBB, ERBB1, HER1
Database cross-references and differences (RAF-indexed):
- Uniprot P00533
- engineered mutation (96)
- engineered mutation (164)
Domains in SCOPe 2.08: d5edpa_
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5edpA (A:)
gsgeapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelreatsp
kankeildeayvmasvdnphvcrllgicltstvqlimqlmpfgclldyvrehkdnigsqy
llnwcvqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfgrakllgaaaaeyhaeg
gkvpikwmalesilhriythqsdvwsygvtvwelmtfgskpydgipaseissilekgerl
pqppictidvymimvkcwmidadsrpkfreliiefskmardpqrylviqgdermhlpspt
dsnfyralmdeedmddvvdadeylipqqgns
Sequence, based on observed residues (ATOM records): (download)
>5edpA (A:)
eapnqallrilketefkkikvlgsgafgtvykglwipegekvkipvaikelatspkanke
ildeayvmasvdnphvcrllgicltstvqlimqlmpfgclldyvrehkdnigsqyllnwc
vqiakgmnyledrrlvhrdlaarnvlvktpqhvkitdfgrakvpikwmalesilhriyth
qsdvwsygvtvwelmtfgskpydgipaseissilekgerlpqppictidvymimvkcwmi
dadsrpkfreliiefskmardpqrylviqgdermhlpsptdsnfddvvdadeyli