PDB entry 5e8x
View 5e8x on RCSB PDB site
Description: tgf-beta receptor type 1 kinase domain (t204d,i211v,y249f,s280t, y282f,s287n,a350c,l352f) in complex with staurosporine
Class: transferase/transferase inhibitor
Keywords: alk5, kinase domain, transferase-transferase inhibitor complex
Deposited on
2015-10-14, released
2016-05-11
The last revision prior to the SCOPe 2.06 freeze date was dated
2016-05-11, with a file datestamp of
2016-05-06.
Experiment type: XRAY
Resolution: 1.45 Å
R-factor: N/A
AEROSPACI score: 0.5
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: TGF-beta receptor type-1
Species: Homo sapiens [TaxId:9606]
Gene: TGFBR1, ALK5, SKR4
Database cross-references and differences (RAF-indexed):
- Uniprot P36897 (3-306)
- engineered mutation (7)
- engineered mutation (14)
- engineered mutation (52)
- engineered mutation (83)
- engineered mutation (85)
- engineered mutation (90)
- engineered mutation (153)
- engineered mutation (155)
Domains in SCOPe 2.06: d5e8xa_ - Heterogens: STU, GOL, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5e8xA (A:)
ghmtiardivlqesvgkgrfgevwrgkwrgeevavkifssreerswfreaeifqtvmlrh
enilgfiaadnkdngtwtqlwlvtdfhehgnlfdylnrytvtvegmiklalstasglahl
hmeivgtqgkpaiahrdlksknilvkkngtccicdfglavrhdsatdtidiapnhrvgtk
rymapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdp
sveemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqls
qqegikm
Sequence, based on observed residues (ATOM records): (download)
>5e8xA (A:)
tiardivlqesvgkgrfgevwrgkwrgeevavkifssreerswfreaeifqtvmlrheni
lgfiaadnkdngtwtqlwlvtdfhehgnlfdylnrytvtvegmiklalstasglahlhme
ivgtqgkpaiahrdlksknilvkkngtccicdfglavrhdsatdtidiapnhrvgtkrym
apevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdpsve
emrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsqqe
gikm