PDB entry 5dp4
View 5dp4 on RCSB PDB site
Description: Crystal Structure of EV71 3C Proteinase in complex with compound 3
Class: hydrolase/hydrolase inhibitor
Keywords: Hand, foot and mouth disease, 3C proteinase, peptidomimetics, drug design, rupintrivir, HYDROLASE-HYDROLASE INHIBITOR complex
Deposited on
2015-09-12, released
2016-03-30
The last revision prior to the SCOPe 2.08 freeze date was dated
2016-04-06, with a file datestamp of
2016-04-01.
Experiment type: XRAY
Resolution: 2.21 Å
R-factor: N/A
AEROSPACI score: 0.25
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: 3C proteinase
Species: ENTEROVIRUS A71 [TaxId:39054]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5dp4a1, d5dp4a2 - Chain 'B':
Compound: 3C proteinase
Species: ENTEROVIRUS A71 [TaxId:39054]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5dp4b1, d5dp4b2 - Chain 'C':
Compound: 3C proteinase
Species: ENTEROVIRUS A71 [TaxId:39054]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5dp4c1, d5dp4c2 - Chain 'D':
Compound: 3C proteinase
Species: ENTEROVIRUS A71 [TaxId:39054]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5dp4d1, d5dp4d2 - Heterogens: 5E8, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5dp4A (A:)
mgpsldfalsllrrnvrqvqtdqghftmlgvrdrlavlprhsqpgktiwiehklvnilda
velvdeqgvnleltlitldtnekfrditkfipenistasdatlvintehmpsmfvpvgdv
vqygflnlsgkpthrtmmynfptkagqcggvvtsvgkvigihiggngrqgfcaglkrsyf
aseqlehhhhhh
Sequence, based on observed residues (ATOM records): (download)
>5dp4A (A:)
mgpsldfalsllrrnvrqvqtdqghftmlgvrdrlavlprhsqpgktiwiehklvnilda
velvdeqgvnleltlitldtnekfrditkfipenistasdatlvintehmpsmfvpvgdv
vqygflnlsgkpthrtmmynfptkagqcggvvtsvgkvigihiggngrqgfcaglkrsyf
a
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5dp4B (B:)
mgpsldfalsllrrnvrqvqtdqghftmlgvrdrlavlprhsqpgktiwiehklvnilda
velvdeqgvnleltlitldtnekfrditkfipenistasdatlvintehmpsmfvpvgdv
vqygflnlsgkpthrtmmynfptkagqcggvvtsvgkvigihiggngrqgfcaglkrsyf
aseqlehhhhhh
Sequence, based on observed residues (ATOM records): (download)
>5dp4B (B:)
mgpsldfalsllrrnvrqvqtdqghftmlgvrdrlavlprhsqpgktiwiehklvnilda
velvdeqgvnleltlitldtnekfrditkfipenistasdatlvintehmpsmfvpvgdv
vqygflnlsgkpthrtmmynfptkagqcggvvtsvgkvigihiggngrqgfcaglkrsyf
a
- Chain 'C':
Sequence, based on SEQRES records: (download)
>5dp4C (C:)
mgpsldfalsllrrnvrqvqtdqghftmlgvrdrlavlprhsqpgktiwiehklvnilda
velvdeqgvnleltlitldtnekfrditkfipenistasdatlvintehmpsmfvpvgdv
vqygflnlsgkpthrtmmynfptkagqcggvvtsvgkvigihiggngrqgfcaglkrsyf
aseqlehhhhhh
Sequence, based on observed residues (ATOM records): (download)
>5dp4C (C:)
mgpsldfalsllrrnvrqvqtdqghftmlgvrdrlavlprhsqpgktiwiehklvnilda
velvdeqgvnleltlitldtnekfrditkfipenistasdatlvintehmpsmfvpvgdv
vqygflnlsgkpthrtmmynfptkagqcggvvtsvgkvigihiggngrqgfcaglkrsyf
a
- Chain 'D':
Sequence, based on SEQRES records: (download)
>5dp4D (D:)
mgpsldfalsllrrnvrqvqtdqghftmlgvrdrlavlprhsqpgktiwiehklvnilda
velvdeqgvnleltlitldtnekfrditkfipenistasdatlvintehmpsmfvpvgdv
vqygflnlsgkpthrtmmynfptkagqcggvvtsvgkvigihiggngrqgfcaglkrsyf
aseqlehhhhhh
Sequence, based on observed residues (ATOM records): (download)
>5dp4D (D:)
mgpsldfalsllrrnvrqvqtdqghftmlgvrdrlavlprhsqpgktiwiehklvnilda
velvdeqgvnleltlitldtnekfrditkfipenistasdatlvintehmpsmfvpvgdv
vqygflnlsgkpthrtmmynfptkagqcggvvtsvgkvigihiggngrqgfcaglkrsyf
a