PDB entry 5d10
View 5d10 on RCSB PDB site
Description: Kinase domain of cSrc in complex with RL236
Class: transferase
Keywords: kinase inhibitor, drug resistance, transferase
Deposited on
2015-08-03, released
2015-09-02
The last revision prior to the SCOPe 2.08 freeze date was dated
2015-09-23, with a file datestamp of
2015-09-18.
Experiment type: XRAY
Resolution: 2.7 Å
R-factor: N/A
AEROSPACI score: 0.17
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Proto-oncogene tyrosine-protein kinase Src
Species: Gallus gallus [TaxId:9031]
Gene: SRC
Database cross-references and differences (RAF-indexed):
- Uniprot P00523 (Start-285)
- engineered mutation (90)
- engineered mutation (97)
Domains in SCOPe 2.08: d5d10a_ - Chain 'B':
Compound: Proto-oncogene tyrosine-protein kinase Src
Species: Gallus gallus [TaxId:9031]
Gene: SRC
Database cross-references and differences (RAF-indexed):
- Uniprot P00523 (Start-285)
- engineered mutation (90)
- engineered mutation (97)
Domains in SCOPe 2.08: d5d10b_ - Heterogens: 563, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5d10A (A:)
ghmqtqglakdaweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaf
lqeaqvmkklrheklvqlyavvseepiyivmeymskgclldflkgemgkylrlpqlvdma
aqiasgmayvermnyvhrdlraanilvgenlvckvadfglarliedneytarqgakfpik
wtapeaalygrftiksdvwsfgilltelttkgrvpypgmvnrevldqvergyrmpcppec
peslhdlmcqcwrkdpeerptfeylqafledyftstepqyqpgenl
Sequence, based on observed residues (ATOM records): (download)
>5d10A (A:)
daweipreslrlevklgqevwmgtwngttrvaiktlkpgtmspeaaqvmkklrheklvql
yavvseepiyivmeymskgclldflkgemgkylrlpqlvdmaaqiasgmayvermnyvhr
dlraanilvgenlvckvadpikwtapeaalygrftiksdvwsfgilltelttkgrvpypg
mvnrevldqvergyrmpcppecpeslhdlmcqcwrkdpeerptfeylqafledyftstep
qyqpgenl
- Chain 'B':
Sequence, based on SEQRES records: (download)
>5d10B (B:)
ghmqtqglakdaweipreslrlevklgqgcfgevwmgtwngttrvaiktlkpgtmspeaf
lqeaqvmkklrheklvqlyavvseepiyivmeymskgclldflkgemgkylrlpqlvdma
aqiasgmayvermnyvhrdlraanilvgenlvckvadfglarliedneytarqgakfpik
wtapeaalygrftiksdvwsfgilltelttkgrvpypgmvnrevldqvergyrmpcppec
peslhdlmcqcwrkdpeerptfeylqafledyftstepqyqpgenl
Sequence, based on observed residues (ATOM records): (download)
>5d10B (B:)
kdaweipreslrlevklgqgcfgevwmgtwngttrvaiktlaqvmkklrheklvqlyavv
seepiyivmeymskgclldflkgemgkylrlpqlvdmaaqiasgmayvermnyvhrdlra
anilvgenlvckvadfglpikwtapeaalygrftiksdvwsfgilltelttkgrvpypgm
vnrevldqvergyrmpcppecpeslhdlmcqcwrkdpeerptfeylqafledyftstepq
yqpgenl