PDB entry 5a00
View 5a00 on RCSB PDB site
Description: Structure of human PARP1 catalytic domain bound to an isoindolinone inhibitor
Class: transferase
Keywords: transferase, human parp1, artd1
Deposited on
2015-04-15, released
2015-08-12
The last revision prior to the SCOPe 2.08 freeze date was dated
2019-03-06, with a file datestamp of
2019-03-01.
Experiment type: XRAY
Resolution: 2.75 Å
R-factor: N/A
AEROSPACI score: 0.17
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Poly [ADP-ribose] polymerase 1
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d5a00a1, d5a00a2 - Heterogens: D7N, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>5a00A (A:)
gpltvnpgtksklpkpvqdlikmifdvesmkkamveyeidlqkmplgklskrqiqaaysi
lsevqqavsqgssdsqildlsnrfytliphdfgmkkppllnnadsvqakvemldnlldie
vaysllrggsddsskdpidvnyeklktdikvvdrdseeaeiirkyvknthatthnaydle
vidifkieregecqrykpfkqlhnrrllwhgsrttnfagilsqglriappeapvtgymfg
kgiyfadmvsksanychtsqgdpiglillgevalgnmyelkhashisklpkgkhsvkglg
kttpdpsanisldgvdvplgtgissgvndtsllyneyivydiaqvnlkyllklkfnfkts
lw
Sequence, based on observed residues (ATOM records): (download)
>5a00A (A:)
ksklpkpvqdlikmifdvesmkkamveyeidlqkmplgklskrqiqaaysilsevqqavs
qgssdsqildlsnrfytliphdppllnnadsvqakvemldnlldievaysllrggskdpi
dvnyeklktdikvvdrdseeaeiirkyvknthatthnaydlevidifkieregecqrykp
fkqlhnrrllwhgsrttnfagilsqglriappeapvtgymfgkgiyfadmvsksanycht
sqgdpiglillgevalgnmyelkhashisklpkgkhsvkglgkttpdpsanisldgvdvp
lgtgissgvndtsllyneyivydiaqvnlkyllklkfnfk