PDB entry 4ylw
View 4ylw on RCSB PDB site
Description: Crystal structure of human dihydroorotate dehydrogenase (DHODH) with No.33 compound
Class: oxidoreductase/oxidoreductase inhibitor
Keywords: Inhibitor, Rheumatoid Arthritis, Complex, OXIDOREDUCTASE-OXIDOREDUCTASE INHIBITOR complex
Deposited on
2015-03-06, released
2016-03-09
The last revision prior to the SCOPe 2.08 freeze date was dated
2016-03-09, with a file datestamp of
2016-03-04.
Experiment type: XRAY
Resolution: 1.79 Å
R-factor: N/A
AEROSPACI score: 0.38
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Dihydroorotate dehydrogenase (quinone), mitochondrial
Species: Homo sapiens [TaxId:9606]
Gene: DHODH
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4ylwa_ - Heterogens: 52Y, FMN, ORO, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4ylwA (A:)
mghhhhhhhhhhssghiddddkhmatgderfyaehlmptlqglldpesahrlavrftslg
llprarfqdsdmlevrvlghkfrnpvgiaagfdkhgeavdglykmgfgfveigsvtpkpq
egnprprvfrlpedqavinrygfnshglsvvehrlrarqqkqakltedglplgvnlgknk
tsvdaaedyaegvrvlgpladylvvnvsspntaglrslqgkaelrrlltkvlqerdglrr
vhrpavlvkiapdltsqdkediasvvkelgidglivtnttvsrpaglqgalrsetgglsg
kplrdlstqtiremyaltqgrvpiigvggvssgqdalekiragaslvqlytaltfwgppv
vgkvkreleallkeqgfggvtdaigadhrr
Sequence, based on observed residues (ATOM records): (download)
>4ylwA (A:)
gderfyaehlmptlqglldpesahrlavrftslgllprarfqdsdmlevrvlghkfrnpv
giaagfdkhgeavdglykmgfgfveigsvtpkpqegnprprvfrlpedqavinrygfnsh
glsvvehrlrarqqkqakltedglplgvnlgknktsvdaaedyaegvrvlgpladylvvn
vsspntaglrslqgkaelrrlltkvlqerdglrrvhrpavlvkiapdltsqdkediasvv
kelgidglivtnttvsrpaglqgalrsetgglsgkplrdlstqtiremyaltqgrvpiig
vggvssgqdalekiragaslvqlytaltfwgppvvgkvkreleallkeqgfggvtdaiga
dhrr