PDB entry 4x2g
View 4x2g on RCSB PDB site
Description: Selection of fragments for kinase inhibitor design: decoration is key
Class: transferase/transferase inhibitor
Keywords: TRANSFERASE, PROTEIN KINASE, INHIBITOR COMPLEX, TRANSFERASE-TRANSFERASE INHIBITOR complex
Deposited on
2014-11-26, released
2015-08-12
The last revision prior to the SCOPe 2.05 freeze date was dated
2015-08-12, with a file datestamp of
2015-08-07.
Experiment type: XRAY
Resolution: 1.51 Å
R-factor: N/A
AEROSPACI score: 0.48
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: TGF-beta receptor type-1
Species: Homo sapiens [TaxId:9606]
Gene: TGFBR1, ALK5, SKR4
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.05: d4x2ga_ - Heterogens: 3WK, SO4, TRS, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4x2gA (A:)
gtiartivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhen
ilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlhm
eivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtkry
mapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdpsv
eemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsqq
egikm
Sequence, based on observed residues (ATOM records): (download)
>4x2gA (A:)
gtiartivlqesigkgrfgevwrgkwrgeevavkifssreerswfreaeiyqtvmlrhen
ilgfiaadnkdngtwtqlwlvsdyhehgslfdylnrytvtvegmiklalstasglahlhm
eivgtqgkpaiahrdlksknilvkkngtcciadlglavrhdsatdtidiapnhrvgtkry
mapevlddsinmkhfesfkradiyamglvfweiarrcsiggihedyqlpyydlvpsdpsv
eemrkvvceqklrpnipnrwqscealrvmakimrecwyangaarltalrikktlsqlsqq
egi