PDB entry 4uyg
View 4uyg on RCSB PDB site
Description: C-Terminal bromodomain of Human BRD2 with I-BET726 (GSK1324726A)
Class: transcription
Keywords: transcription, inhibitor, histone, epigenetic reader, bet, brd2
Deposited on
2014-08-31, released
2014-10-08
The last revision prior to the SCOPe 2.08 freeze date was dated
2014-10-22, with a file datestamp of
2014-10-17.
Experiment type: XRAY
Resolution: 2.5 Å
R-factor: 0.19249
AEROSPACI score: 0.27
(click here for full SPACI score report)
Chains and heterogens:
- Chain 'A':
Compound: Bromodomain-containing protein 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4uyga_ - Chain 'B':
Compound: Bromodomain-containing protein 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4uygb_ - Chain 'C':
Compound: Bromodomain-containing protein 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4uygc_ - Chain 'D':
Compound: Bromodomain-containing protein 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4uygd_ - Chain 'E':
Compound: Bromodomain-containing protein 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4uyge_ - Chain 'F':
Compound: Bromodomain-containing protein 2
Species: Homo sapiens [TaxId:9606]
Database cross-references and differences (RAF-indexed):
Domains in SCOPe 2.08: d4uygf_ - Heterogens: 73B, SO4, HOH
PDB Chain Sequences:
- Chain 'A':
Sequence, based on SEQRES records: (download)
>4uygA (A:)
mgsshhhhhhssglvprgshmhqsskkgklseqlkhcngilkellskkhaayawpfykpv
dasalglhdyhdiikhpmdlstvkrkmenrdyrdaqefaadvrlmfsncykynppdhdvv
amarklqdvfefryakmpdeplepgplpvstamppgl
Sequence, based on observed residues (ATOM records): (download)
>4uygA (A:)
seqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmenr
dyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
- Chain 'B':
Sequence, based on SEQRES records: (download)
>4uygB (B:)
mgsshhhhhhssglvprgshmhqsskkgklseqlkhcngilkellskkhaayawpfykpv
dasalglhdyhdiikhpmdlstvkrkmenrdyrdaqefaadvrlmfsncykynppdhdvv
amarklqdvfefryakmpdeplepgplpvstamppgl
Sequence, based on observed residues (ATOM records): (download)
>4uygB (B:)
seqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmenr
dyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
- Chain 'C':
Sequence, based on SEQRES records: (download)
>4uygC (C:)
mgsshhhhhhssglvprgshmhqsskkgklseqlkhcngilkellskkhaayawpfykpv
dasalglhdyhdiikhpmdlstvkrkmenrdyrdaqefaadvrlmfsncykynppdhdvv
amarklqdvfefryakmpdeplepgplpvstamppgl
Sequence, based on observed residues (ATOM records): (download)
>4uygC (C:)
gklseqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkm
enrdyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
- Chain 'D':
Sequence, based on SEQRES records: (download)
>4uygD (D:)
mgsshhhhhhssglvprgshmhqsskkgklseqlkhcngilkellskkhaayawpfykpv
dasalglhdyhdiikhpmdlstvkrkmenrdyrdaqefaadvrlmfsncykynppdhdvv
amarklqdvfefryakmpdeplepgplpvstamppgl
Sequence, based on observed residues (ATOM records): (download)
>4uygD (D:)
eqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmenrd
yrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
- Chain 'E':
Sequence, based on SEQRES records: (download)
>4uygE (E:)
mgsshhhhhhssglvprgshmhqsskkgklseqlkhcngilkellskkhaayawpfykpv
dasalglhdyhdiikhpmdlstvkrkmenrdyrdaqefaadvrlmfsncykynppdhdvv
amarklqdvfefryakmpdeplepgplpvstamppgl
Sequence, based on observed residues (ATOM records): (download)
>4uygE (E:)
seqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmenr
dyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd
- Chain 'F':
Sequence, based on SEQRES records: (download)
>4uygF (F:)
mgsshhhhhhssglvprgshmhqsskkgklseqlkhcngilkellskkhaayawpfykpv
dasalglhdyhdiikhpmdlstvkrkmenrdyrdaqefaadvrlmfsncykynppdhdvv
amarklqdvfefryakmpdeplepgplpvstamppgl
Sequence, based on observed residues (ATOM records): (download)
>4uygF (F:)
lseqlkhcngilkellskkhaayawpfykpvdasalglhdyhdiikhpmdlstvkrkmen
rdyrdaqefaadvrlmfsncykynppdhdvvamarklqdvfefryakmpd