PDB entry 4uez

View 4uez on RCSB PDB site
Description: Crystal structure of the human CARBOXYPEPTIDASE A1 in complex with the PHOSPHINIC INHIBITOR Acetyl-Leu-Phe-Y(PO2CH2)-Phe-OH
Class: hydrolase
Keywords: hydrolase, carboxypeptidase, cpa1, phosphinic inhibitor
Deposited on 2014-12-22, released 2016-01-20
The last revision prior to the SCOPe 2.08 freeze date was dated 2016-01-20, with a file datestamp of 2016-01-15.
Experiment type: XRAY
Resolution: 2.29 Å
R-factor: N/A
AEROSPACI score: 0.25 (click here for full SPACI score report)

Chains and heterogens:

  • Chain 'A':
    Compound: human carboxypeptidase a1
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d4ueza_
  • Chain 'B':
    Compound: human carboxypeptidase a1
    Species: Homo sapiens [TaxId:9606]
    Database cross-references and differences (RAF-indexed): Domains in SCOPe 2.08: d4uezb_
  • Heterogens: ZN, LFF, HOH

PDB Chain Sequences:

  • Chain 'A':
    Sequence, based on SEQRES records: (download)
    >4uezA (A:)
    arstdtfnyatyhtleeiydfldllvaenphlvskiqigntyegrpiyvlkfstggskrp
    aiwidtgihsrewvtqasgvwfakkitqdygqdaaftaildtldifleivtnpdgfafth
    stnrmwrktrshtagslcigvdpnrnwdagfglsgassnpcsetyhgkfansevevksiv
    dfvkdhgnikafisihsysqllmypygyktepvpdqdeldqlskaavtalaslygtkfny
    gsiikaiyqasgstidwtysqgikysftfelrdtgrygfllpasqiiptaketwlallti
    mehtlnhpy
    

    Sequence, based on observed residues (ATOM records): (download)
    >4uezA (A:)
    stdtfnyatyhtleeiydfldllvaenphlvskiqigntyegrpiyvlkfstggskrpai
    widtgihsrewvtqasgvwfakkitqdygqdaaftaildtldifleivtnpdgfafthst
    nrmwrktrshtagslcigvdpnrnwdagfglsgassnpcsetyhgkfansevevksivdf
    vkdhgnikafisihsysqllmypygyktepvpdqdeldqlskaavtalaslygtkfnygs
    iikaiyqasgstidwtysqgikysftfelrdtgrygfllpasqiiptaketwlalltime
    htlnhp
    

  • Chain 'B':
    Sequence, based on SEQRES records: (download)
    >4uezB (B:)
    arstdtfnyatyhtleeiydfldllvaenphlvskiqigntyegrpiyvlkfstggskrp
    aiwidtgihsrewvtqasgvwfakkitqdygqdaaftaildtldifleivtnpdgfafth
    stnrmwrktrshtagslcigvdpnrnwdagfglsgassnpcsetyhgkfansevevksiv
    dfvkdhgnikafisihsysqllmypygyktepvpdqdeldqlskaavtalaslygtkfny
    gsiikaiyqasgstidwtysqgikysftfelrdtgrygfllpasqiiptaketwlallti
    mehtlnhpy
    

    Sequence, based on observed residues (ATOM records): (download)
    >4uezB (B:)
    rstdtfnyatyhtleeiydfldllvaenphlvskiqigntyegrpiyvlkfstggskrpa
    iwidtgihsrewvtqasgvwfakkitqdygqdaaftaildtldifleivtnpdgfafths
    tnrmwrktrshtagslcigvdpnrnwdagfglsgassnpcsetyhgkfansevevksivd
    fvkdhgnikafisihsysqllmypygyktepvpdqdeldqlskaavtalaslygtkfnyg
    siikaiyqasgstidwtysqgikysftfelrdtgrygfllpasqiiptaketwlalltim
    ehtlnhp